SCHEMBL5548901

SCHEMBL5548901

CC(Nc1nc(C(C)(C)C)cn2c(=O)[nH]nc12)C(O)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.38
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CHRM2 P08172 1/20 0.35
ADRA1A P35348 1/20 0.35
RGS12 O14924 1/20 0.35
GLA P06280 1/20 0.35
CYP2D6 P10635 1/20 0.35
PKM P14618 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
ALOX12 P18054 1/20 0.35
ADRA2C P18825 1/20 0.35
NFKB1 P19838 1/20 0.35
HTR2A P28223 1/20 0.35
CYP2C19 P33261 1/20 0.35
THPO P40225 1/20 0.35
GNAI1 P63096 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PDE5A O76074 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5550127 0.87 CYP3A4 (0.37) CYP3A4CYP2C9PDE5AKMT2AMEN1
SCHEMBL5548550 0.77 NTRK1 (0.39) CYP2C9PDE5A
SCHEMBL3524781 0.71 CLK4 (0.45) GLAPDE5AKMT2AMEN1KDM4E
SCHEMBL5545590 0.71 GSK3B (0.35)
SCHEMBL5549383 0.71 MAPT (0.40) CYP3A4ADRA1ACYP2D6ALOX15TSHR
SCHEMBL5545469 0.69 ADORA1 (0.41) HSD17B10KMT2AMEN1KDM4ELMNA
SCHEMBL5549023 0.69 ADORA1 (0.38) CYP3A4CYP2C9TSHRCYP2C19HSD17B10
SCHEMBL5549142 0.68 GSK3B (0.35)
SCHEMBL3528837 0.68 GSK3B (0.47)
SCHEMBL5545525 0.68 ADORA1 (0.47) NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed