SCHEMBL5549023

SCHEMBL5549023

CC(C)(C)c1cn2c(=O)[nH]nc2c(NCc2cccc3ccccc23)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.38
PIK3CB P42338 5/20 0.38
BRDT Q58F21 1/20 0.38
SOS1 Q07889 1/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
BRD4 O60885 1/20 0.37
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
AURKB Q96GD4 1/20 0.36
PIK3CA P42336 3/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CG P48736 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 1/20 0.35
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5549030 0.83 THRB (0.40) ADORA1ALDH1A1LMNAMAPTMEN1
SCHEMBL3528837 0.79 GSK3B (0.47) ADORA1
SCHEMBL3523080 0.78 GSK3A (0.50) ADORA1ALDH1A1LMNAMAPTMEN1
SCHEMBL5549007 0.78 KMT2A (0.51) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL5543068 0.78 SMN1; SMN2 (0.41) ADORA1ALDH1A1LMNAMAPTMEN1
SCHEMBL5545434 0.77 GPR18 (0.46) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL5545643 0.77 GSK3B (0.34) ADORA1
SCHEMBL5550039 0.77 GSK3A (0.46) ADORA1LMNAMAPTMEN1KMT2A
SCHEMBL5545556 0.76 GSK3A (0.48) ADORA1
SCHEMBL5543587 0.76 GSK3B (0.39) ADORA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed