SCHEMBL5550190

SCHEMBL5550190

NC(=O)c1ccc(N2CCN(C(=O)Cc3ccc4ccccc4c3)CC2)nc1CCc1cccc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
BTK Q06187 1/20 0.41
GFER P55789 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GPR183 P32249 1/20 0.40
ME2 P23368 1/20 0.40
ME1 P48163 1/20 0.40
ME3 Q16798 1/20 0.40
PANK3 Q9H999 3/20 0.40
GBA1 P04062 1/20 0.38
ADRB2 P07550 1/20 0.38
KCNH2 Q12809 1/20 0.38
GRM5 P41594 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5586271 0.82 SCD (0.46) KMT2AKDM4EALDH1A1HPGDME2
SCHEMBL3669356 0.76 NPC1 (0.51) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL3676046 0.70 SCD (0.54) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL9320601 0.69 MEN1 (0.68) ATMMEN1KMT2AGFERKDM4E
SCHEMBL9410731 0.68 GPR183 (0.56) ATMMEN1KMT2AGFERALDH1A1
SCHEMBL11077598 0.68 ATM (0.51) ATMMEN1KMT2AKDM4EALDH1A1
SCHEMBL10911138 0.67 POLB (0.68) ATMMEN1KMT2AALDH1A1
SCHEMBL11081503 0.67 KDM4E (0.62) KDM4EALDH1A1HPGDHSD17B10GPR183
SCHEMBL24095043 0.66 ADRB2 (0.73) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL24095122 0.66 ADRB2 (0.76) ATMMEN1KMT2AALDH1A1ME2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763350-A1 NICOTINAMIDE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-03-21 EP disclosed
WO-2006014168-A1 NICOTINAMIDE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2006-02-09 WO disclosed