SCHEMBL5552192

SCHEMBL5552192

CCc1n[nH]c(CN)c1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 7/20 0.43
DPP4 P27487 2/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRB2 P47870 1/20 0.34
GABRA4 P48169 1/20 0.34
GABRE P78334 1/20 0.34
GABRA6 Q16445 1/20 0.34
GABRG1 Q8N1C3 1/20 0.34
GABRG3 Q99928 1/20 0.34
GABRQ Q9UN88 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11203864 0.84 HCAR2 (0.44) HCAR2GABRPGABRDGABRA1GABRB1
SCHEMBL11210298 0.79 HCAR2 (0.41) HCAR2GABRPGABRDGABRA1GABRB1
SCHEMBL12486045 0.74 HCAR2 (0.42) HCAR2TTRP2RX7NPC1RAB9A
SCHEMBL27737815 0.72 HCAR2 (0.54) HCAR2DPP4GABRPGABRDGABRA1
SCHEMBL2077234 0.72 HCAR2 (0.52) HCAR2GABRPGABRDGABRA1GABRB1
SCHEMBL9218944 0.69 HCAR2 (0.43) HCAR2DPP4DPP8DPP9TTR
SCHEMBL3804253 0.67 GAA (0.40) HCAR2GABRPGABRDGABRA1GABRB1
Hydrochloric Acid SCHEMBL5287806 0.66 P2RX7 (0.36) HCAR2TTRP2RX7
SCHEMBL3402262 0.66 P2RX7 (0.48) HCAR2DPP4DPP9TTRP2RX7
SCHEMBL27737480 0.65 HCAR2 (0.49) HCAR2GABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781661-A2 VASOPRESSIN V1A ANTAGONISTS Ferring B.V. (NL) 2007-05-09 EP disclosed
WO-2006021213-A2 VASOPRESSIN V1A ANTAGONISTS FERRING B.V. (NL) 2006-03-02 WO disclosed