SCHEMBL555290

SCHEMBL555290

CCCCOC(=O)/C=C/C(=O)OC

nearest known ligand 0.83

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.83
HCAR2 Q8TDS4 7/20 0.71
MAPT P10636 1/20 0.66
RAB9A P51151 1/20 0.66
NPSR1 Q6W5P4 1/20 0.66
HPGD P15428 1/20 0.59
TSHR P16473 1/20 0.59
KEAP1 Q14145 1/20 0.54
NFE2L2 Q16236 1/20 0.54
ALDH1A1 P00352 1/20 0.50
APP P05067 5/20 0.47
EPHX1 P07099 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2302656 1.00 ATM (0.83) ATMHCAR2MAPTRAB9ANPSR1
Dimethyl Maleate SCHEMBL8992612 1.00 ATM (0.83) ATMHCAR2MAPTRAB9ANPSR1
Dimethyl Fumarate SCHEMBL8992615 1.00 ATM (0.83) ATMHCAR2MAPTRAB9ANPSR1
SCHEMBL2302660 1.00 ATM (0.83) ATMHCAR2MAPTRAB9ANPSR1
SCHEMBL22619937 0.96 ATM (0.77) ATMHCAR2MAPTRAB9ANPSR1
SCHEMBL10389785 0.94 ATM (0.73) ATMHCAR2MAPTRAB9ANPSR1
SCHEMBL554181 0.94 ATM (0.73) ATMHCAR2MAPTRAB9ANPSR1
Monomethyl Fumarate SCHEMBL28123679 0.93 HCAR2 (0.86) ATMHCAR2MAPTRAB9ANPSR1
Butyl Fumarate SCHEMBL9358646 0.93 HCAR2 (0.86) ATMHCAR2MAPTRAB9ANPSR1
Butyl Fumarate SCHEMBL9358650 0.93 HCAR2 (0.86) ATMHCAR2MAPTRAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 166 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022186442-A1 PRESSURE-SENSITIVE ADHESIVE COMPOSITION WITH EXCELLENT PIGMENT DISPERSIBILITY, AND PRESSURE-SENSITIVE ADHESIVE SHEET USING SAME 주식회사 켐코 2022-09-09 WO claimed
US-20220105064-A1 CONTROLLED RELEASE PHARMACEUTICAL COMPOSITIONS COMPRISING A FUMARIC ACID ESTER BIOGEN SWISS MFG GMBH (CH) 2022-04-07 US claimed
US-20220079884-A1 PHARMACEUTICAL FORMULATION COMPRISING ONE OR MORE FUMARIC ACID ESTERS IN AN EROSION MATRIX BIOGEN SWISS MFG GMBH (CH) 2022-03-17 US claimed
US-11229619-B2 Controlled release pharmaceutical compositions comprising a fumaric acid ester BIOGEN SWISS MANUFACTURING GMBH (CH) 2022-01-25 US claimed
US-20180221284-A1 PHARMACEUTICAL FORMULATION COMPRISING ONE OR MORE FUMARIC ACID ESTERS IN AN EROSION MATRIX BIOGEN SWISS MANUFACTURING GMBH (CH) 2018-08-09 US claimed
US-20150272894-A1 PHARMACEUTICAL FORMULATION COMPRISING ONE OR MORE FUMARIC ACID ESTERS IN AN EROSION MATRIX BIOGEN SWISS MANUFACTURING GMBH (CH) 2015-10-01 US claimed
US-20130259906-A1 PHARMACEUTICAL COMPOSITION COMPRISING ONE OR MORE FUMARIC ACID ESTERS FORWARD PHARMA A/S (DK) 2013-10-03 US claimed
US-20120034303-A1 PHARMACEUTICAL FORMULATION COMPRISING ONE OR MORE FUMARIC ACID ESTERS IN AN EROSION MATRIX FORWARD PHARMA A/S (DK) 2012-02-09 US claimed
US-20120034274-A1 PHARMACEUTICAL COMPOSITION COMPRISING ONE OR MORE FUMARIC ACID ESTERS FORWARD PHARMA A/S (DK) 2012-02-09 US claimed
EP-2379062-A1 PHARMACEUTICAL COMPOSITION COMPRISING ONE OR MORE FUMARIC ACID ESTERS Forward Pharma A/S (DK) 2011-10-26 EP claimed
EP-2379063-A1 PHARMACEUTICAL FORMULATION COMPRISING ONE OR MORE FUMARIC ACID ESTERS IN AN EROSION MATRIX Forward Pharma A/S (DK) 2011-10-26 EP claimed
WO-2010079222-A1 PHARMACEUTICAL FORMULATION COMPRISING ONE OR MORE FUMARIC ACID ESTERS IN AN EROSION MATRIX FORWARD PHARMA A/S (DK) 2010-07-15 WO claimed
WO-2010079221-A1 PHARMACEUTICAL COMPOSITION COMPRISING ONE OR MORE FUMARIC ACID ESTERS FORWARD PHARMA A/S (DK) 2010-07-15 WO claimed
WO-2025089083-A1 GAS-BARRIER LAMINATE AND PACKAGING MATERIAL DIC株式会社 2025-05-01 WO disclosed
US-20250026928-A1 CROSSLINKABLE RESIN COMPOSITION, CURED PRODUCT, LAMINATE AND HEAT-RESISTANT MEMBER DIC CORPORATION (JP) 2025-01-23 US disclosed
US-20250010592-A1 GAS BARRIER FILM AND PACKAGING MATERIAL DIC CORPORATION (JP) 2025-01-09 US disclosed
EP-1165488-A1 PROCESS FOR THE PREPARATION OF POLYAMINO SUCCINIC ACIDS AND DERIVATIVES THEREOF THE DOW CHEMICAL COMPANY (US) 2002-01-02 EP disclosed
US-20010034300-A1 Reacting an alpha, beta unsaturated carboxylic acid ester with a heterocyclic oxygen nitrogen, or sulfur compound NIPPON SHOKUBAI COMPANY LTD. (JP) 2001-10-25 US disclosed
EP-1123915-A1 Process for producing alpha, beta-unsaturated carboxylic acid esters and catalyst for use in such process Nippon Shokubai Co., Ltd. (JP) 2001-08-16 EP disclosed
WO-2000058263-A1 PROCESS FOR THE PREPARATION OF POLYAMINO SUCCINIC ACIDS AND DERIVATIVES THEREOF THE DOW CHEMICAL COMPANY (US) 2000-10-05 WO disclosed