Butyl Fumarate

Butyl Fumarate

SCHEMBL9358646

CCCCOC(=O)/C=C\C(=O)O.COC(=O)/C=C\C(=O)O

nearest known ligand 0.86

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KEAP1

The experimentally established mechanism targets of Butyl Fumarate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KEAP1 known ✓ Q14145 1/20 0.46
HCAR2 Q8TDS4 8/20 0.86
ATM Q13315 1/20 0.71
MAPT P10636 3/20 0.58
RAB9A P51151 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
HPGD P15428 1/20 0.52
TSHR P16473 1/20 0.52
NFE2L2 Q16236 1/20 0.46
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 2/20 0.45
TDP1 Q9NUW8 1/20 0.45
APP P05067 2/20 0.43
ALOX15 P16050 1/20 0.42
RECQL P46063 1/20 0.42
HSD17B10 Q99714 1/20 0.42
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Butyl Fumarate SCHEMBL9358650 1.00 HCAR2 (0.86) HCAR2ATMMAPTRAB9ANPSR1
Monomethyl Fumarate SCHEMBL28123679 1.00 HCAR2 (0.86) HCAR2ATMMAPTRAB9ANPSR1
Butyl Fumarate SCHEMBL1655582 0.93 HCAR2 (0.92) HCAR2ATMMAPTRAB9ANPSR1
Butyl Fumarate SCHEMBL27358297 0.93 HCAR2 (1.00) HCAR2ATMMAPTRAB9ANPSR1
Butyl Fumarate SCHEMBL124163 0.93 HCAR2 (1.00) HCAR2ATMMAPTRAB9ANPSR1
Butyl Fumarate SCHEMBL4376900 0.93 HCAR2 (1.00) HCAR2ATMMAPTRAB9ANPSR1
Butyl Fumarate SCHEMBL43165 0.93 HCAR2 (1.00) HCAR2ATMMAPTRAB9ANPSR1
Butyl Fumarate SCHEMBL43164 0.93 HCAR2 (1.00) HCAR2ATMMAPTRAB9ANPSR1
Maleic Acid SCHEMBL28199237 0.93 HCAR2 (1.00) HCAR2ATMMAPTRAB9ANPSR1
Butyl Fumarate SCHEMBL29604195 0.93 HCAR2 (1.00) HCAR2ATMMAPTRAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0285140-B1 Process for producing toner for developing electrostatic images CANON KK (JP) 1994-12-21 EP disclosed
US-4839255-A IMPACTING MODIFIER TO BASE PARTICLES CANON KABUSHIKI KAISHA (JP) 1989-06-13 US disclosed
EP-0285140-A2 Process for producing toner for developing electrostatic images CANON KABUSHIKI KAISHA (JP) 1988-10-05 EP disclosed