SCHEMBL5553550

SCHEMBL5553550

CCc1[nH]c(-c2cccc3ccccc23)nc1C=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 1/20 0.39
PI4K2B Q8TCG2 1/20 0.39
PI4K2A Q9BTU6 1/20 0.39
PI4KB Q9UBF8 1/20 0.39
MAPK13 O15264 1/20 0.38
GCGR P47871 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
BCHE P06276 1/20 0.35
KDM4E B2RXH2 2/20 0.35
IDO1 P14902 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
GUSB P08236 1/20 0.35
ALOX5 P09917 1/20 0.35
TYMS P04818 1/20 0.35
ALOX15 P16050 2/20 0.35
PPARG P37231 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963578 0.83 NPC1 (0.45) KDM4EGAA
SCHEMBL5549123 0.80 MAPK13 (0.44) PI4KAPI4K2BPI4K2API4KBMAPK13
SCHEMBL5552730 0.77 KDM4E (0.43) PI4KAPI4K2BPI4K2API4KBKDM4E
SCHEMBL5554927 0.73 KDM4E (0.48) KDM4ECYP1A2ALOX15
SCHEMBL3404703 0.70 PI4KA (0.45) PI4KAPI4K2BPI4K2API4KBMAPK13
SCHEMBL186872 0.69 PI4KA (0.49) PI4KAPI4K2BPI4K2API4KBMAPK13
SCHEMBL30516197 0.68 TYMP (0.50) PI4KAPI4K2BPI4K2API4KBMAPK13
SCHEMBL24317556 0.68 PI4KA (0.47) PI4KAPI4K2BPI4K2API4KBMAPK13
SCHEMBL415342 0.66 KDM4E (0.46) PI4KAPI4K2BPI4K2API4KBMAPK13
SCHEMBL27729265 0.66 PI4KA (0.47) PI4KAPI4K2BPI4K2API4KBMAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848428-A2 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORPORATION (US) 2007-10-31 EP disclosed
WO-2006089076-A2 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORPORATION (US) 2006-08-24 WO disclosed