SCHEMBL5554095

SCHEMBL5554095

COc1ccc2c(c1)c(OC(C)=O)c(C)n2C(=O)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.56
AKR1C2 P52895 6/20 0.56
PPARG P37231 6/20 0.51
PPARA Q07869 3/20 0.51
PTGS2 P35354 3/20 0.51
LMNA P02545 2/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2D6 P10635 2/20 0.51
CYP2C9 P11712 2/20 0.51
HIF1A Q16665 2/20 0.51
NPSR1 Q6W5P4 2/20 0.51
PTGS1 P23219 2/20 0.51
TSHR P16473 1/20 0.51
NFKB1 P19838 1/20 0.51
KDM4E B2RXH2 1/20 0.51
MEN1 O00255 1/20 0.51
PTGES O14684 1/20 0.51
ABCC3 O15438 1/20 0.51
ABCC4 O15439 1/20 0.51
ABCB11 O95342 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5554001 0.89 PTGS1 (0.46) AKR1C3AKR1C2PPARGPPARAPTGS2
SCHEMBL5822660 0.88 AKR1C3 (0.65) AKR1C3AKR1C2PPARGPTGS2LMNA
SCHEMBL1076364 0.86 PTGS2 (0.65) AKR1C3AKR1C2PPARGPTGS2LMNA
SCHEMBL8579955 0.85 LMNA (0.65) AKR1C3AKR1C2PPARGPTGS2LMNA
SCHEMBL11436509 0.85 PTGS2 (0.64) AKR1C3AKR1C2PPARGPTGS2LMNA
SCHEMBL5797468 0.84 AKR1C3 (0.52) AKR1C3AKR1C2PPARGPTGS2LMNA
Water SCHEMBL11448360 0.84 PTGS2 (0.62) AKR1C3AKR1C2PPARGPTGS2LMNA
Water SCHEMBL11448358 0.84 PTGS2 (0.62) AKR1C3AKR1C2PPARGPTGS2LMNA
SCHEMBL5558979 0.83 AKR1C3 (0.39) AKR1C3AKR1C2PPARGPPARA
SCHEMBL5799148 0.82 PTGS2 (0.52) AKR1C3AKR1C2PPARGPTGS2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed