SCHEMBL5555174

SCHEMBL5555174

CCOC(=O)COc1ccc(C(Br)C(=O)OC)cc1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.55
NPSR1 Q6W5P4 1/20 0.55
PTPN1 P18031 1/20 0.49
POLB P06746 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46
MAPT P10636 2/20 0.46
ALDH1A1 P00352 1/20 0.46
TP53 P04637 1/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.44
LMNA P02545 1/20 0.44
TBXAS1 P24557 1/20 0.44
MAPK1 P28482 1/20 0.44
EPHX2 P34913 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20484981 0.86 ACACB (0.50) GAANPSR1POLBSMN1; SMN2ALDH1A1
SCHEMBL5556095 0.85 SMN1; SMN2 (0.50) PTPN1SMN1; SMN2MAPTMAPK1
SCHEMBL6577434 0.84 GAA (0.59) GAANPSR1PTPN1POLBSMN1; SMN2
SCHEMBL5551276 0.83 LTA4H (0.48) SMN1; SMN2MAPTMAPK1
SCHEMBL6185341 0.81 TAS1R3 (0.51) SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL9000712 0.81 SMN1; SMN2 (0.57) POLBSMN1; SMN2KDM4ELMNAMAPK1
SCHEMBL2624372 0.80 GAA (0.62) GAANPSR1PTPN1POLBKDM4E
SCHEMBL12742268 0.79 GAA (0.57) GAANPSR1PTPN1POLBSMN1; SMN2
SCHEMBL435444 0.78 GAA (0.68) GAANPSR1PTPN1POLBSMN1; SMN2
SCHEMBL11815554 0.78 GAA (0.72) GAANPSR1PTPN1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1301750-C Conjugates of macrocyclic metal complexes with biomolucules and utilization thereof for producing agents for use in NMR diagnosis and radiodiagnosis and radiotherapy SCHERING AG (DE) 2007-02-28 CN disclosed
US-20070014725-A1 Conjugates of macrocyclic metal complexes with biomolecules and their use for the production of agents for NMR diagnosis and radiodiagnosis as well as radiotherapy SCHERING AG (DE) 2007-01-18 US disclosed
US-7164016-B2 Macrocyclic metal complexes and their use for the production of conjugates with biomolecules SCHERING AG (DE) 2007-01-16 US disclosed
US-20070009442-A1 Macrocyclic metal complexes and their use for the production of conjugates with biomolecules SCHERING AG (DE) 2007-01-11 US disclosed
CN-1541114-A Conjugates of macrocyclic metal complexes with biomolucules and utilization thereof for producing agents for use in NMR diagnosis and radiodiagnosis and radiotherapy ���ֹɷݹ�˾ 2004-10-27 CN disclosed
CN-1533286-A Macrocyclic metal complexes and use thereof for production of conjugates with biomolecules ���ֹɷݹ�˾ 2004-09-29 CN disclosed
US-20030206865-A1 Conjugates of macrocyclic metal complexes with biomolecules and their use for the production of agents for NMR diagnosis and radiodiagnosis as well as radiotherapy SCHERING AG (DE) 2003-11-06 US disclosed
US-20030108486-A1 Macrocyclic metal complexes and their use for the production of conjugates with biomolecules SCHERING AG (DE) 2003-06-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030108486-A1 Macrocyclic metal complexes and their use for the production of conjugates with biomolecules CA13, MPI, CA14 GAA 814/4885NPSR1 1305/4885PTPN1 4741/4885
US-20070014725-A1 Conjugates of macrocyclic metal complexes with biomolecules and their use for the production of agents for NMR diagnosis and radiodiagnosis as well as radiotherapy CA13, CA14, CA12 GAA 754/4885NPSR1 1976/4885PTPN1 4824/4885
US-20030206865-A1 Conjugates of macrocyclic metal complexes with biomolecules and their use for the production of agents for NMR diagnosis and radiodiagnosis as well as radiotherapy CA13, CA14, CA12 GAA 754/4885NPSR1 1976/4885PTPN1 4824/4885
US-20070009442-A1 Macrocyclic metal complexes and their use for the production of conjugates with biomolecules CA13, MPI, CA14 GAA 814/4885NPSR1 1305/4885PTPN1 4741/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.