SCHEMBL5555837

SCHEMBL5555837

CCc1c(CC(=O)NC)nn(C(C)C)c1Oc1cccc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP2C9 P11712 1/20 0.38
OGG1 O15527 1/20 0.37
HRH3 Q9Y5N1 2/20 0.36
MGLL Q99685 1/20 0.36
SLC6A4 P31645 2/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HTT P42858 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5562406 0.90 CARM1 (0.33) PTGDR2
SCHEMBL5555927 0.84 CYP1A2 (0.40) PTGER4CYP1A2CYP2C19CYP2C9OGG1
SCHEMBL5562003 0.84 CYP1A2 (0.38) PTGER4CYP1A2CYP2C19CYP2C9OGG1
SCHEMBL5564780 0.83 OGG1 (0.38) PTGER4CYP1A2CYP2C19CYP2C9OGG1
SCHEMBL5561559 0.83 CYP1A2 (0.38) PTGER4CYP1A2CYP2C19CYP2C9OGG1
SCHEMBL5561153 0.82 CYP1A2 (0.40) PTGER4CYP1A2CYP2C19CYP2C9OGG1
SCHEMBL5559739 0.81 CYP1A2 (0.43) PTGER4CYP1A2CYP2C19CYP2C9OGG1
SCHEMBL5561125 0.80 MEN1 (0.37) KMT2AHTTLMNANPSR1FNTA
SCHEMBL5556106 0.80 CYP1A2 (0.40) PTGER4CYP1A2CYP2C19CYP2C9OGG1
SCHEMBL5561735 0.78 MAPT (0.37) CYP1A2CYP2C19KMT2AL3MBTL1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597235-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-08-15 EP disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed