SCHEMBL5556285

SCHEMBL5556285

CCC(C)OC(=O)C(C)c1c(C)n(C(=O)c2ccc(Cl)c(F)c2)c2cc(F)c(O)cc12

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.36
PTGS2 P35354 9/20 0.33
PTGS1 P23219 1/20 0.33
AKR1C3 P42330 2/20 0.32
AKR1C2 P52895 2/20 0.32
IDO1 P14902 1/20 0.32
KCNH2 Q12809 1/20 0.32
ABCB1 P08183 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5814808 0.92 MGLL (0.34) MGLLPTGS2AKR1C3AKR1C2
SCHEMBL5559475 0.91 PTGS2 (0.41) PTGS2PTGS1AKR1C3AKR1C2ABCB1
SCHEMBL6426560 0.91 PTGS2 (0.41) PTGS2PTGS1AKR1C3AKR1C2ABCB1
SCHEMBL5809718 0.91 PTGS2 (0.36) PTGS2PTGS1AKR1C3AKR1C2ABCB1
SCHEMBL5809713 0.91 PTGS2 (0.36) PTGS2PTGS1AKR1C3AKR1C2ABCB1
SCHEMBL5822684 0.89 PTGS2 (0.43) PTGS2PTGS1AKR1C3AKR1C2
SCHEMBL5801106 0.88 MGLL (0.41) MGLL
SCHEMBL5814796 0.88 PTGS2 (0.38) PTGS2PTGS1AKR1C3AKR1C2
SCHEMBL5814801 0.88 PTGS2 (0.38) PTGS2PTGS1AKR1C3AKR1C2
SCHEMBL5813349 0.86 PTGS2 (0.40) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed