SCHEMBL5560309

SCHEMBL5560309

Cc1c(CC(=O)O)c2cc(OC(=O)C(c3c(C)n(C(=O)c4cccc(F)c4)c4cc(F)c(O)cc34)C3CCC3)c(F)cc2n1C(=O)c1cccc(F)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 6/20 0.44
AKR1C2 P52895 6/20 0.44
PTGIR P43119 9/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
HIF1A Q16665 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PTGS1 P23219 2/20 0.39
PTGS2 P35354 2/20 0.39
PTGDR Q13258 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5798238 0.86 AKR1C3 (0.48) AKR1C3AKR1C2PTGIRLMNACYP1A2
SCHEMBL5798161 0.85 AKR1C3 (0.46) AKR1C3AKR1C2PTGIRLMNACYP1A2
SCHEMBL5797739 0.85 AKR1C3 (0.45) AKR1C3AKR1C2PTGIRLMNACYP1A2
SCHEMBL6427504 0.84 USP2 (0.39) AKR1C3AKR1C2LMNA
SCHEMBL6425674 0.82 TDP1 (0.41) AKR1C3AKR1C2LMNA
SCHEMBL5559087 0.82 AKR1C3 (0.62) AKR1C3AKR1C2LMNACYP1A2CYP2D6
SCHEMBL5560429 0.77 PTGS1 (0.45) AKR1C3AKR1C2PTGIRLMNACYP1A2
SCHEMBL5800814 0.76 AKR1C3 (0.48) AKR1C3AKR1C2LMNACYP1A2CYP2D6
SCHEMBL6423088 0.76 ALDH1A1 (0.37)
SCHEMBL5800291 0.76 LMNA (0.39) AKR1C3AKR1C2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed