SCHEMBL5560838

SCHEMBL5560838

CC(C)n1nc(CO)c(Cc2ccncc2)c1Oc1cccc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.39
PDE4B Q07343 2/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RHEB Q15382 1/20 0.35
PSEN1 P49768 4/20 0.35
PSEN2 P49810 4/20 0.35
APH1B Q8WW43 4/20 0.35
NCSTN Q92542 4/20 0.35
APH1A Q96BI3 4/20 0.35
PSENEN Q9NZ42 4/20 0.35
TRPC5 Q9UL62 2/20 0.35
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
FLT1 P17948 2/20 0.34
KDR P35968 2/20 0.34
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5560726 0.87 CYP1A2 (0.41) CYP1A2CYP2C9CYP2C19RHEBPSEN1
SCHEMBL5562261 0.87 L3MBTL1 (0.39) PDE4DPDE4BCYP1A2CYP2C9CYP2C19
SCHEMBL5555927 0.85 CYP1A2 (0.40) CYP1A2CYP2C9CYP2C19RHEBPSEN1
SCHEMBL5556169 0.80 CYP1A2 (0.44) CYP1A2CYP2C9CYP2C19RHEBPSEN1
SCHEMBL5562098 0.79 CYP1A2 (0.38) CYP1A2CYP2C9CYP2C19ALDH1A1MAPT
SCHEMBL5208321 0.78 PDE4D (0.36) PDE4DPDE4BKMT2AL3MBTL1ALDH1A1
SCHEMBL14453961 0.77 PSEN1 (0.39) CYP1A2CYP2C9CYP2C19KMT2ARHEB
SCHEMBL5562173 0.75 EPAS1 (0.34) CYP1A2CYP2C19
SCHEMBL5561153 0.74 CYP1A2 (0.40) CYP1A2CYP2C9CYP2C19RHEBPSEN1
SCHEMBL14471402 0.73 ROCK2 (0.40) PDE4DPDE4BKMT2AL3MBTL1RHEB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597235-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-08-15 EP disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed
US-7241794-B2 Nonnucleoside reverse transcriptase inhibitors ROCHEPALO ALTO LLC (US) 2007-07-10 US disclosed