SCHEMBL5567280

SCHEMBL5567280

Cc1ccc(C(=O)NC2CC2)cc1-c1ccc2c(cnn2-c2ccccc2)n1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KHK P50053 3/20 0.55
MAPK14 Q16539 9/20 0.54
MAPK11 Q15759 2/20 0.54
RIPK2 O43353 7/20 0.53
LCK P06239 2/20 0.49
KIT P10721 2/20 0.49
KDR P35968 2/20 0.49
CYP2C9 P11712 1/20 0.49
MAPK13 O15264 1/20 0.48
RAF1 P04049 1/20 0.48
PDGFRA P16234 1/20 0.48
MAPKAPK2 P49137 1/20 0.48
MAPK12 P53778 1/20 0.48
KCNH2 Q12809 1/20 0.48
HPGDS O60760 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2216662 0.85 KHK (0.57) KHKMAPK14MAPK11RIPK2LCK
SCHEMBL2214287 0.78 KHK (0.54) KHKMAPK14MAPK11RIPK2LCK
SCHEMBL4229997 0.75 NR3C1 (0.58) MAPK14MAPK11RIPK2LCKKIT
SCHEMBL2214290 0.73 MAPK14 (0.54) KHKMAPK14MAPK11RIPK2LCK
SCHEMBL2216168 0.73 MAPK14 (0.66) MAPK14MAPK11RIPK2LCKKIT
SCHEMBL4219336 0.72 HPGDS (0.55) KHKMAPK14CYP2C9MAPK13HPGDS
SCHEMBL31367847 0.72 MAPK14 (0.74) MAPK14MAPK11RIPK2LCKKIT
SCHEMBL3519858 0.72 MAPK14 (0.82) MAPK14MAPK11MAPK13MAPK12
SCHEMBL4219489 0.72 NR3C1 (0.56) MAPK14MAPK11RIPK2LCKKIT
SCHEMBL23711737 0.71 KHK (1.00) KHKMAPK14MAPK11HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070161673-A1 P38 kinase inhibitors SMITHKLINE BEECHAM CORPORATION 2007-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070161673-A1 P38 kinase inhibitors MAPK1, MAPK7, MAP3K1 KHK 2805/4885MAPK14 14/4885MAPK11 38/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.