SCHEMBL5568415

SCHEMBL5568415

CC[C@H](N)C(=O)N1c2ccccc2C[C@@H]1OC(=O)NCC1CC1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
MTNR1A P48039 3/20 0.40
MTNR1B P49286 3/20 0.40
DRD2 P14416 1/20 0.40
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6240896 0.89 KDM4E (0.57) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL6242771 0.88 KDM4E (0.60) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL6244892 0.86 KDM4E (0.55) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL6242475 0.86 KDM4E (0.70) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5568632 0.85 KDM4E (0.52) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL6242776 0.85 KDM4E (0.60) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5563867 0.84 KDM4E (0.54) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5563916 0.82 KDM4E (0.74) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
Trifluoroacetic Acid SCHEMBL5569107 0.77 KDM4E (0.65) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5568600 0.73 ALDH1A1 (0.42) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042288-B1 TRIPEPTIDYL PEPTIDASE INHIBITORS INST NAT SANTE RECH MED (FR) 2007-11-07 EP claimed