SCHEMBL5568477

SCHEMBL5568477

Cc1cc(C)c(N(CCN(C)C)S(=O)(=O)c2cc(Cl)cc(Cl)c2OC(=O)NCc2c(NS(=O)(=O)c3cc(Cl)cc(Cl)c3O)cccc2N2CCCCC2)c(C)c1N1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACLY P53396 16/20 0.39
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
HPGD P15428 1/20 0.34
MCOLN2 Q8IZK6 1/20 0.33
KDM4E B2RXH2 2/20 0.32
GAA P10253 2/20 0.32
XBP1 P17861 1/20 0.32
HTT P42858 1/20 0.32
PAX8 Q06710 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ACACB O00763 1/20 0.32
ACACA Q13085 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL534166 0.79 ACLY (0.39) ACLYALDH1A1LMNAKDM4E
SCHEMBL8313576 0.78 ACLY (0.52) ACLYMEN1KMT2AALDH1A1LMNA
SCHEMBL533013 0.77 ACLY (0.53) ACLYMEN1KMT2ALMNAMAPT
SCHEMBL534072 0.74 ACLY (0.36) ACLYMEN1KMT2AALDH1A1LMNA
SCHEMBL532938 0.70 ACLY (0.55) ACLYMEN1KMT2ALMNAMAPT
SCHEMBL533484 0.70 ACLY (0.58) ACLYMAPTACACBACACA
SCHEMBL533060 0.69 ACLY (0.52) ACLYMEN1KMT2AACACBACACA
SCHEMBL533015 0.68 ACLY (0.54) ACLY
SCHEMBL533530 0.67 ALDH1A1 (0.39) MEN1KMT2AALDH1A1LMNAMAPT
SCHEMBL5566597 0.67 ACLY (0.40) ACLYMEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1610753-A4 PHENYLENEDIAMINE UROTENSIN-II RECEPTOR ANTAGONISTS AND CCR-9 ANTAGONISTS ENCYSIVE PHARMACEUTICALS INC (US) 2007-07-04 EP disclosed
EP-1610753-A2 PHENYLENEDIAMINE UROTENSIN-II RECEPTOR ANTAGONISTS AND CCR-9 ANTAGONISTS ENCYSIVE PHARMACEUTICALS INC. (US) 2006-01-04 EP disclosed
WO-2004073634-A2 PHENYLENEDIAMINE UROTENSIN-II RECEPTOR ANTAGONISTS AND CCR-9 ANTAGONISTS ENCYSIVE PHARMACEUTICALS INC. (US) 2004-09-02 WO disclosed