SCHEMBL5569182

SCHEMBL5569182

CC1(C)CC1(CN)c1ccc(C(=O)NCCC(=O)Nc2ccc(Cl)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.53
ALDH1A1 P00352 1/20 0.53
RHOC P08134 2/20 0.50
RHOA P61586 2/20 0.50
RAB9A P51151 1/20 0.49
CYP1A2 P05177 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
MAOB P27338 1/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
BLM P54132 1/20 0.45
PMP22 Q01453 1/20 0.45
MAPT P10636 1/20 0.44
EPHX2 P34913 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5567044 0.86 RAB9A (0.61) POLBALDH1A1RAB9ACYP1A2TSHR
SCHEMBL5569181 0.79 POLB (0.55) POLBALDH1A1RHOCRHOARAB9A
SCHEMBL5566675 0.78 POLB (0.57) POLBALDH1A1RHOCRHOARAB9A
SCHEMBL5569234 0.78 POLB (0.55) POLBALDH1A1RHOCRHOARAB9A
SCHEMBL5570403 0.77 ALDH1A1 (0.54) POLBALDH1A1RHOCRHOARAB9A
SCHEMBL5569176 0.77 POLB (0.53) POLBALDH1A1RHOCRHOARAB9A
SCHEMBL5566055 0.73 ALDH1A1 (0.52) POLBALDH1A1RHOCRHOARAB9A
SCHEMBL5629014 0.69 POLB (0.55) POLBALDH1A1RHOCRHOARAB9A
SCHEMBL16527695 0.67 IDO1 (0.54) POLBALDH1A1RHOCRHOARAB9A
SCHEMBL16542660 0.67 IDO1 (0.60) POLBALDH1A1RHOCRHOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7250415-B2 1,1-Disubstitutedcycloalkyl-, glycinamidyl-, sulfonyl-amidino-, and tetrahydropyrimidinyl-containing diaminoalkyl, β-aminoacids, α-aminoacids and derivatives thereof as factor Xa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-07-31 US disclosed