SCHEMBL5569424

SCHEMBL5569424

CCCCNC(=O)[C@H]1Cc2cc(OC)ccc2N1C(=O)[C@@H](N)CC

nearest known ligand 0.72

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.72
CYP2D6 P10635 2/20 0.72
KDM4E B2RXH2 1/20 0.72
CYP1A2 P05177 1/20 0.72
CYP3A4 P08684 1/20 0.72
TDP1 Q9NUW8 1/20 0.72
MAPT P10636 1/20 0.47
LMNA P02545 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6247284 0.91 ALDH1A1 (0.59) ALDH1A1CYP2D6KDM4ECYP1A2CYP3A4
SCHEMBL6243667 0.91 ALDH1A1 (0.59) ALDH1A1CYP2D6KDM4ECYP1A2CYP3A4
SCHEMBL6242188 0.90 ALDH1A1 (0.57) ALDH1A1CYP2D6KDM4ECYP1A2CYP3A4
Oxalic Acid SCHEMBL7043586 0.89 KDM4E (0.56) ALDH1A1CYP2D6KDM4ECYP1A2CYP3A4
Oxalic Acid SCHEMBL7043599 0.89 KDM4E (0.56) ALDH1A1CYP2D6KDM4ECYP1A2CYP3A4
SCHEMBL6240391 0.87 KDM4E (0.76) ALDH1A1CYP2D6KDM4ECYP1A2CYP3A4
SCHEMBL6247072 0.87 KDM4E (0.76) ALDH1A1CYP2D6KDM4ECYP1A2CYP3A4
SCHEMBL5569373 0.87 KDM4E (0.76) ALDH1A1CYP2D6KDM4ECYP1A2CYP3A4
Oxalic Acid SCHEMBL7041574 0.87 ALDH1A1 (0.55) ALDH1A1CYP2D6KDM4ECYP1A2CYP3A4
SCHEMBL5568469 0.86 KDM4E (0.74) ALDH1A1CYP2D6KDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042288-B1 TRIPEPTIDYL PEPTIDASE INHIBITORS INST NAT SANTE RECH MED (FR) 2007-11-07 EP disclosed
US-6335360-B1 INDOLINE-2-CARBOXYLIC AMIDE DERIVATIVES; OBESITY, EATING AND PSYCHOLOGICAL DISORDERS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2002-01-01 US disclosed