SCHEMBL5575014

SCHEMBL5575014

COc1cc2nc(-c3ccc(-c4ccccc4)c(F)c3)nc(Nc3ccc4c(cnn4C(=O)O)c3)c2cc1OC(C)=O

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 16/20 0.44
ROCK2 O75116 2/20 0.43
ABCB1 P08183 9/20 0.42
ABCC1 P33527 4/20 0.42
ERBB2 P04626 1/20 0.42
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL877185 0.92 EGFR (0.44) ABCG2ROCK2ABCB1ABCC1ERBB2
SCHEMBL878022 0.91 ABCG2 (0.45) ABCG2ABCB1ABCC1ERBB2MEN1
SCHEMBL877263 0.89 ERBB2 (0.47) ABCG2ROCK2ABCB1ABCC1ERBB2
SCHEMBL877621 0.87 ROCK2 (0.45) ABCG2ROCK2ABCB1ABCC1ERBB2
SCHEMBL877821 0.84 ROCK2 (0.45) ABCG2ROCK2ABCB1ABCC1ERBB2
SCHEMBL876652 0.84 ABCG2 (0.57) ABCG2ABCB1MEN1POLBMAPT
SCHEMBL876653 0.84 ABCG2 (0.57) ABCG2ABCB1MEN1POLBMAPT
SCHEMBL877259 0.83 EGFR (0.45) ABCG2ROCK2ABCB1ABCC1ERBB2
SCHEMBL877820 0.83 ROCK2 (0.54) ABCG2ROCK2ERBB2MEN1MAPT
SCHEMBL877683 0.82 EGFR (0.44) ABCG2ROCK2ABCB1ABCC1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1865958-A2 PHARMACOKINETICALLY IMPROVED COMPOUNDS Surface Logix, Inc. (US) 2007-12-19 EP disclosed
WO-2006105081-A2 PHARMACOKINETICALLY IMPROVED COMPOUNDS SURFACE LOGIX, INC. (US) 2006-10-05 WO disclosed