SCHEMBL878022

SCHEMBL878022

COc1cc2nc(-c3ccc(-c4ccccc4)c(F)c3)nc(Nc3ccc4c(cnn4C(=O)O)c3)c2cc1O

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 17/20 0.45
ABCB1 P08183 9/20 0.43
ABCC1 P33527 4/20 0.43
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
SYK P43405 1/20 0.41
ERBB2 P04626 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL877259 0.92 EGFR (0.45) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL5575014 0.91 ABCG2 (0.44) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL877746 0.91 ABCG2 (0.48) ABCG2ABCB1ABCC1ERBB2
SCHEMBL877263 0.89 ERBB2 (0.47) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL877747 0.89 ABCG2 (0.43) ABCG2ABCB1ABCC1MEN1LMNA
SCHEMBL877745 0.89 ABCG2 (0.49) ABCG2ABCB1ABCC1ERBB2
SCHEMBL1724776 0.84 ROCK2 (0.44) ABCG2ABCB1ABCC1SYKERBB2
SCHEMBL877294 0.84 ABCG2 (0.58) ABCG2ABCB1MEN1MAPTKMT2A
SCHEMBL877293 0.84 ABCG2 (0.58) ABCG2ABCB1MEN1MAPTKMT2A
SCHEMBL877185 0.83 EGFR (0.44) ABCG2ABCB1ABCC1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012040499-A2 METABOLIC INHIBITORS SURFACE LOGIX, INC. (US) 2012-03-29 WO disclosed