SCHEMBL5577183

SCHEMBL5577183

COc1c(C=O)cc(Cl)cc1N1CCN(C(C)(C)C)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.39
MAPT P10636 1/20 0.39
ERN1 O75460 3/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HTR1A P08908 3/20 0.36
DRD2 P14416 3/20 0.36
DRD4 P21917 3/20 0.36
HTR2A P28223 3/20 0.36
HTR2C P28335 3/20 0.36
DRD3 P35462 3/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 3/20 0.34
ALDH1A3 P47895 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4931500 0.82 MEN1 (0.44) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL27422458 0.71 HTR3E (0.64) ALDH1A1MAPTDRD2DRD4LMNA
SCHEMBL1748175 0.70 ERN1 (0.66) ALDH1A1ERN1MEN1KMT2AHPGD
SCHEMBL14292141 0.70 ERN1 (0.51) ALDH1A1ERN1MEN1KMT2AHPGD
SCHEMBL27250826 0.69 ATR (0.37) MAPTLMNAHTR3EHTR3BHTR3A
SCHEMBL30925338 0.69 ATR (0.37) MAPTLMNAHTR3EHTR3BHTR3A
SCHEMBL6413771 0.68 ERN1 (0.53) ALDH1A1ERN1MEN1KMT2AHPGD
SCHEMBL31551028 0.68 ERN1 (0.53) ALDH1A1ERN1MEN1KMT2AHPGD
SCHEMBL5577210 0.67 NPSR1 (0.34) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL415808 0.67 ERN1 (0.51) ALDH1A1MAPTERN1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1750727-A2 KINASE MODULATORS AND METHODS OF USE Exelixis, Inc. (US) 2007-02-14 EP disclosed
WO-2005117909-A2 KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2005-12-15 WO disclosed