SCHEMBL5577313

SCHEMBL5577313

Cc1c(Br)cc(C(=O)Nc2ccccc2)cc1N1CCN(C(C)(C)C)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
TP53 P04637 3/20 0.43
MAPT P10636 2/20 0.43
RPS6KB1 P23443 1/20 0.42
AKT1 P31749 1/20 0.42
HTR1D P28221 3/20 0.42
HTR1B P28222 3/20 0.42
HTR2A P28223 3/20 0.42
RBP4 P02753 1/20 0.41
CNR1 P21554 2/20 0.41
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 2/20 0.41
POLB P06746 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CHRM1 P11229 1/20 0.40
CNR2 P34972 1/20 0.40
GAA P10253 1/20 0.39
KMT2A Q03164 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4932179 0.85 PTPN11 (0.52) MAPTRBP4ALDH1A1KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL4931665 0.83 POLB (0.46) TP53MAPTRPS6KB1AKT1HTR1D
SCHEMBL2301569 0.75 AKT1 (0.59) RPS6KB1AKT1P2RY12
SCHEMBL2454605 0.70 MAPT (0.68) NPC1RAB9ATP53MAPTSMN1; SMN2
SCHEMBL12644447 0.68 HSPD1 (0.64) TP53MAPTALDH1A1KMT2APLG
SCHEMBL10245047 0.67 KDM4E (0.65) MAPTRBP4ALDH1A1KDM4EHPGD
SCHEMBL14043612 0.67 NPC1 (0.75) NPC1RAB9ATP53MAPTCNR1
SCHEMBL2911616 0.65 HDAC2 (0.71) NPC1RAB9AKDM4EHPGDPOLB
SCHEMBL11589882 0.65 HSPD1 (0.64) TP53MAPTALDH1A1KMT2APLG
SCHEMBL19382960 0.65 L3MBTL1 (0.60) NPC1RAB9AMAPTPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1750727-A2 KINASE MODULATORS AND METHODS OF USE Exelixis, Inc. (US) 2007-02-14 EP disclosed
WO-2005117909-A2 KINASE MODULATORS AND METHODS OF USE EXELIXIS, INC. (US) 2005-12-15 WO disclosed