SCHEMBL5577409

SCHEMBL5577409

CN(C)c1ccc(CN2CC=C(c3cccc(CNC(=O)c4ccc(F)cc4)c3)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.63
NPSR1 Q6W5P4 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
CHRM3 P20309 8/20 0.50
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
HTR1A P08908 2/20 0.47
TP53 P04637 1/20 0.45
THRB P10828 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HTT P42858 1/20 0.45
LMNA P02545 1/20 0.44
TNF P01375 1/20 0.44
NOD2 Q9HC29 1/20 0.44
NOD1 Q9Y239 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5577772 0.93 KDM4E (0.54) MAPK1CHRM3MEN1KMT2AHTR1A
SCHEMBL5577708 0.92 CHRM3 (0.54) MAPK1CHRM3MEN1KMT2AHTR1A
SCHEMBL5577268 0.90 CHRM3 (0.49) MAPK1CHRM3MEN1KMT2ATP53
SCHEMBL5577472 0.90 CHRM3 (0.58) MAPK1CHRM3MEN1KMT2ATP53
SCHEMBL5577404 0.90 CHRM3 (0.50) MAPK1CHRM3TP53THRBKDM4E
SCHEMBL5577813 0.89 CHRM3 (0.58) MAPK1CHRM3TP53
SCHEMBL5577388 0.88 CHRM3 (0.60) CHRM3MEN1KMT2AHTR1ATHRB
SCHEMBL5577540 0.87 CHRM3 (0.51) MAPK1NPSR1TDP1CHRM3MEN1
SCHEMBL5577397 0.85 ALDH1A1 (0.55) CHRM3MEN1KMT2AALDH1A1
SCHEMBL5577436 0.84 MAPK1 (0.50) MAPK1NPSR1TDP1CHRM3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070043079-A1 Heterocyclic compound containing nitrogen atom and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-02-22 US disclosed
EP-1616862-A1 NITROGENOUS HETEROCYCLIC COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2006-01-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070043079-A1 Heterocyclic compound containing nitrogen atom and use thereof HLA-DRB1, MIF, HLA-C MAPK1 592/4885NPSR1 235/4885TDP1 3686/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.