SCHEMBL5577688

SCHEMBL5577688

Cc1c(Cl)cccc1C(=O)NCc1ccccc1N1CCN(Cc2ccc(F)cc2)CC1C

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MT-CO2 P00403 4/20 0.48
DRD2 P14416 3/20 0.42
DRD3 P35462 1/20 0.42
GNRHR P30968 1/20 0.41
DRD4 P21917 2/20 0.41
TP53 P04637 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
NR3C1 P04150 1/20 0.40
CCR1 P32246 1/20 0.40
TOP1 P11387 1/20 0.39
CCR5 P51681 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5577655 0.87 S1PR1 (0.45) DRD2DRD3DRD4LMNA
SCHEMBL5577919 0.87 MT-CO2 (0.52) MT-CO2TP53CCR1TOP1CCR5
SCHEMBL5577376 0.87 MAPK8 (0.43) MT-CO2TP53NR3C1CCR1
SCHEMBL5577302 0.85 MT-CO2 (0.48) MT-CO2TOP1CCR5LMNA
SCHEMBL5577730 0.84 CCR1 (0.48) DRD2DRD3GNRHRDRD4CCR1
SCHEMBL5577489 0.83 MT-CO2 (0.48) MT-CO2DRD2DRD3GNRHRTP53
SCHEMBL5577826 0.83 MT-CO2 (0.49) MT-CO2DRD2DRD3
SCHEMBL5577911 0.82 MT-CO2 (0.45) MT-CO2CCR1TOP1LMNA
SCHEMBL5577671 0.82 MT-CO2 (0.43) MT-CO2DRD3SIGMAR1CCR1TOP1
SCHEMBL5577507 0.82 MT-CO2 (0.50) MT-CO2DRD2DRD3DRD4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070043079-A1 Heterocyclic compound containing nitrogen atom and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-02-22 US disclosed
EP-1616862-A1 NITROGENOUS HETEROCYCLIC COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2006-01-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070043079-A1 Heterocyclic compound containing nitrogen atom and use thereof HLA-DRB1, MIF, HLA-C MT-CO2 2047/4885DRD2 4468/4885DRD3 4080/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.