SCHEMBL5580334

SCHEMBL5580334

Cc1ccccc1NC(=O)C(=O)Cl

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.77
RAB9A P51151 2/20 0.77
HPGD P15428 5/20 0.62
ALDH1A1 P00352 2/20 0.62
POLB P06746 2/20 0.56
KDM4E B2RXH2 2/20 0.55
GAA P10253 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
ALOX12 P18054 1/20 0.53
PDK1 Q15118 1/20 0.53
PDK2 Q15119 1/20 0.53
PDK3 Q15120 1/20 0.53
PDK4 Q16654 1/20 0.53
MAPT P10636 2/20 0.53
PLA2G1B P04054 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2344209 0.87 NPC1 (1.00) NPC1RAB9AHPGDALDH1A1POLB
SCHEMBL31411480 0.87 NPC1 (1.00) NPC1RAB9AHPGDALDH1A1POLB
SCHEMBL1270302 0.83 RAB9A (0.69) NPC1RAB9AHPGDALDH1A1POLB
SCHEMBL6857852 0.82 NPC1 (0.88) NPC1RAB9AHPGDALDH1A1POLB
SCHEMBL3723177 0.82 RAB9A (0.80) NPC1RAB9AHPGDALDH1A1POLB
SCHEMBL30852954 0.82 RAB9A (0.80) NPC1RAB9AHPGDALDH1A1POLB
SCHEMBL10780666 0.80 NPC1 (0.65) NPC1RAB9AHPGDALDH1A1POLB
SCHEMBL25356036 0.80 NPC1 (0.77) NPC1RAB9AHPGDALDH1A1POLB
SCHEMBL959541 0.80 NPC1 (0.77) NPC1RAB9AHPGDALDH1A1POLB
SCHEMBL8006309 0.80 NPC1 (0.77) NPC1RAB9AHPGDALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116751151-B One-pot method for preparing 5-chloro-7-methyl isatin 瑞弘(天津)科技有限公司 2025-10-10 CN disclosed
US-7276511-B2 Benzylamine derivative ZERIA PHARMACEUTICAL CO., LTD. (JP) 2007-10-02 US disclosed
US-20060194841-A1 E.g., N-{2-(3,4-dichlorophenyl)-2-[(3,3-diphenylpropionyl)-methylamino]-4-{spiro[benzo(c)thiophene-1(3H),4'-piperidine]-(2S)-oxide}-1'-yl-butyl}-3,3,3-trifluoro-N-methyl-propionamide hydrochloride, NK-1 or NK-2 receptor antagonists; irritable bowel syndrome, pain, anxiety, COPD, headaches and vomiting ZERIA PHARMACEUTICAL CO., LTD. (JP) 2006-08-31 US disclosed
EP-1650189-A1 BENZYLAMINE DERIVATIVE Zeria Pharmaceutical Co., Ltd. (JP) 2006-04-26 EP disclosed
US-6117885-A Biphenyl-substituted quinoline derivatives E. R. SQUIBB & SONS, INC. (US) 2000-09-12 US disclosed
EP-0556060-A1 Biphenyl-substituted quinoline and naphthyridines derivatives as angiotensine II antagonists E.R. SQUIBB & SONS, INC. (US) 1993-08-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060194841-A1 E.g., N-{2-(3,4-dichlorophenyl)-2-[(3,3-diphenylpropionyl)-methylamino]-4-{spiro[benzo(c)thiophene-1(3H),4'-piperidine]-(2S)-oxide}-1'-yl-butyl}-3,3,3-trifluoro-N-methyl-propionamide hydrochloride, NK-1 or NK-2 receptor antagonists; irritable bowel syndrome, pain, anxiety, COPD, headaches and vomiting KCNAB1, BDKRB2, ARRB1 NPC1 386/4885RAB9A 1811/4885HPGD 690/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.