SCHEMBL5581822

SCHEMBL5581822

N#CC(O)c1ccc[nH]1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967495 0.78
SCHEMBL11153273 0.78 MCL1 (0.33)
SCHEMBL29838200 0.77 MCL1 (0.39)
SCHEMBL27343778 0.75
SCHEMBL5094060 0.74
SCHEMBL10833402 0.74
SCHEMBL10366551 0.74 DAO (0.37)
SCHEMBL4409393 0.74
SCHEMBL28764956 0.71 MCL1 (0.34)
SCHEMBL5698996 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7300784-B2 Nitrile hydratase and a method for producing amides DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2007-11-27 US disclosed
US-6900037-B2 Method for producing amide compounds DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2005-05-31 US disclosed
US-20040209345-A1 Nitrile Hydratase and a Method for Producing Amides DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2004-10-21 US disclosed
US-20030124691-A1 Method for producing amide compounds DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2003-07-03 US disclosed
EP-1266962-A2 Method for producing amide compounds Daicel Chemical Industries, Ltd. (JP) 2002-12-18 EP disclosed
EP-0666320-B1 Process for producing alpha-hydroxy acid or alpha-hydroxyamide by microorganisms MITSUBISHI RAYON CO (JP) 2000-12-20 EP disclosed
EP-0711836-B1 Method of producing optically active alpha-hydroxy acid or alpha-hydroxyamide MITSUBISHI RAYON CO (JP) 2000-02-02 EP disclosed
US-5756306-A HYDROLYSIS OF COMPOUNDS USING MICROORGAMISMS TO FORM ALPHA HYDROXY ACIDS OR AMIDES NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1998-05-26 US disclosed
US-5736385-A NITRILASE OR NITRILE HYDRATASE HYDROLYSIS OF A CYANOHYDRIN WHILE AUTOMATICALLY CONTROLLING CYANOHYDRIN CONCENTRATION NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1998-04-07 US disclosed
EP-0773297-A2 Process for producing alfa-hydroxy acid or alfa-hydroxyamide by microorganism NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1997-05-14 EP disclosed
EP-0711836-A1 Method of producing optically active alpha-hydroxy acid or alpha-hydroxyamide NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1996-05-15 EP disclosed
US-5508181-A REACTING AN ALPHA-HYDROXYNITRILE (OR MIXTURE WITH AN ALDEHYDE) WITH HYDROGEN CYANIDE IN PRESENCE OF PHOSPHITE OR HYPOPHOSPHITE IONS NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1996-04-16 US disclosed
EP-0666320-A2 Process for producing alpha-hydroxy acid or alpha-hydroxyamide by microorganisms NITTO CHEMICAL INDUSTRY CO., LTD. (JP) 1995-08-09 EP disclosed