SCHEMBL5586035

SCHEMBL5586035

NC(=O)c1ccc2c(c1)ON=CC2

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
KDM1A O60341 2/20 0.37
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
CASP3 P42574 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
LCK P06239 1/20 0.35
HTR1A P08908 1/20 0.35
HTR1D P28221 1/20 0.35
HTR2C P28335 1/20 0.35
PARP1 P09874 5/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HSD17B3 P37058 1/20 0.33
CHEK2 O96017 2/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9995987 0.87 TSHR (0.47) TSHRKDM1ANPC1RAB9ACASP3
SCHEMBL19207342 0.85 ALDH1A1 (0.46) TSHRKDM4EALDH1A1MAPK1
Carbamic Acid SCHEMBL6649969 0.73 HSD17B10 (0.34) TSHRNPC1RAB9APARP1KDM4E
SCHEMBL3712693 0.72 TDP1 (0.46) TSHRRAB9AKDM4EALDH1A1MAPK1
SCHEMBL6649924 0.72 TSHR (0.49) TSHRKDM1ANPC1RAB9ACASP3
SCHEMBL10509462 0.71 NPC1 (0.46) NPC1RAB9AKDM4E
Hydrochloric Acid SCHEMBL10700892 0.71 TDP1 (0.45) TSHRRAB9AKDM4EALDH1A1MAPK1
SCHEMBL4320180 0.69 TSHR (0.68) TSHRKDM1ANPC1RAB9ACASP3
SCHEMBL30344379 0.69 TSHR (0.68) TSHRKDM1ANPC1RAB9ACASP3
SCHEMBL5125994 0.68 CA12 (0.41) TSHRRAB9AALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740584-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105802-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed