SCHEMBL5586397

SCHEMBL5586397

CC1(c2ccc(C=O)cc2)CCNC1=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.36
CYP2A6 P11509 3/20 0.35
PTGER3 P43115 5/20 0.33
ALDH1A1 P00352 4/20 0.32
TYR P14679 1/20 0.32
CYP2A13 Q16696 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
HSD17B10 Q99714 1/20 0.31
ALDH5A1 P51649 1/20 0.31
ABAT P80404 1/20 0.31
ALDH3A1 P30838 1/20 0.31
ALDH1A3 P47895 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27035682 0.79 CYP19A1 (0.57) CYP19A1
SCHEMBL27229513 0.79 GRIN1 (0.49) CYP19A1PTGER3ALDH1A1GRIN1GRIN2A
SCHEMBL22147812 0.79 GRIN1 (0.49) CYP19A1PTGER3ALDH1A1GRIN1GRIN2A
SCHEMBL23516613 0.73 TYR (0.44) CYP2A6ALDH1A1TYRCYP2A13ALDH1A3
SCHEMBL20914690 0.72 LPL (0.41) CYP19A1
SCHEMBL5177793 0.70 CYP2A6 (0.46) CYP2A6ALDH1A1TYRCYP2A13HSD17B10
SCHEMBL21848155 0.70 GRIN1 (0.40) CYP19A1PTGER3GRIN1GRIN2AGRIN2B
SCHEMBL30683300 0.70 CYP19A1 (0.37) CYP19A1PTGER3GRIN1GRIN2AGRIN2B
SCHEMBL27035700 0.70 CYP19A1 (0.37) CYP19A1PTGER3GRIN1GRIN2AGRIN2B
SCHEMBL2308698 0.69 GRIN1 (0.53) PTGER3GRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8168658-B2 Inhibitors of histone deacetylase MERCK SHARP & DOHME CORP. (US) 2012-05-01 US disclosed
US-20090069250-A1 Inhibitors of Histone Deacetylase MERCK SHARP & DOHME LLC 2009-03-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090069250-A1 Inhibitors of Histone Deacetylase HDAC1, HDAC5, HDAC6 CYP19A1 2145/4885CYP2A6 3249/4885PTGER3 2180/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.