SCHEMBL5591398

SCHEMBL5591398

Cc1ccc(-c2csc(NC(=O)c3cnc(N4CCNC(C(=O)O)C4)c(Cl)c3)n2)cc1C

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MPL P40238 14/20 0.66
NPC1 O15118 2/20 0.43
MEN1 O00255 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
POLB P06746 1/20 0.42
ABL1 P00519 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5590976 0.85 MPL (0.66) MPL
SCHEMBL5591267 0.82 MPL (0.56) MPLNPC1MEN1RAB9AKMT2A
SCHEMBL5591050 0.82 MPL (0.57) MPLNPC1MEN1RAB9AKMT2A
SCHEMBL5590838 0.81 MPL (0.65) MPL
SCHEMBL5591118 0.80 MPL (0.74) MPLABL1
SCHEMBL5591145 0.80 MPL (1.00) MPL
SCHEMBL5591002 0.79 MPL (0.81) MPL
SCHEMBL5591168 0.78 MPL (0.81) MPL
SCHEMBL5590857 0.74 MPL (0.61) MPLABL1
SCHEMBL5591212 0.74 MPL (0.84) MPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007004038-A1 AMINOTHIAZOLE DERIVATIVES AS AGONISTS OF THE THROMBOPOIETIN RECEPTOR PFIZER PRODUCTS INC. (US) 2007-01-11 WO claimed
WO-2007004038-A1 AMINOTHIAZOLE DERIVATIVES AS AGONISTS OF THE THROMBOPOIETIN RECEPTOR PFIZER PRODUCTS INC. (US) 2007-01-11 WO disclosed