SCHEMBL5591850

SCHEMBL5591850

FC(F)(F)c1cccc2sc(-c3ccccc3)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.44
TNF P01375 1/20 0.42
NOD1 Q9Y239 1/20 0.42
ESR1 P03372 1/20 0.42
NR1H2 P55055 1/20 0.42
NR1H3 Q13133 1/20 0.42
ADORA3 P0DMS8 2/20 0.41
ADORA2A P29274 2/20 0.41
ADORA1 P30542 2/20 0.41
AKR1B1 P15121 1/20 0.41
MAPT P10636 4/20 0.40
KDM4E B2RXH2 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 2/20 0.40
GLA P06280 2/20 0.40
GAA P10253 2/20 0.40
PKM P14618 2/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27678949 0.87 TNF (0.49) APPTNFNOD1ADORA3ADORA2A
SCHEMBL5591881 0.84 RAB9A (0.55) MAPTKDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL900790 0.78 ALDH1A1 (0.56) APPADORA3ADORA2AADORA1MAPT
SCHEMBL2137814 0.78 SMN1; SMN2 (0.56) APPADORA3ADORA2AADORA1MAPT
SCHEMBL9314321 0.78 APP (0.44) APPADORA3ADORA2AADORA1MAPT
SCHEMBL900779 0.77 ALDH1A1 (0.47) MAPTKDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL24818889 0.76 ALDH1A1 (0.40) AKR1B1MAPTKDM4ESMN1; SMN2MEN1
SCHEMBL22891113 0.76 ALDH1A1 (0.43) AKR1B1MAPTKDM4ESMN1; SMN2MEN1
SCHEMBL28215029 0.76 APP (0.45) APPADORA3ADORA2AADORA1MAPT
SCHEMBL27856621 0.75 PDCD1 (0.41) ADORA3ADORA2AADORA1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115057830-A Method for synthesizing 2-aryl benzothiazole 辽宁科技大学 2022-09-16 CN disclosed
WO-2007076104-A1 VANILLOID RECEPTOR LIGANDS AND THEIR USE IN TREATMENTS AMGEN INC. (US) 2007-07-05 WO disclosed
EP-1585726-A1 FUSED HETEROCYCLIC DERIVATIVES AS PPAR MODULATORS ELI LILLY AND COMPANY (US) 2005-10-19 EP disclosed
WO-2004063155-A1 FUSED HETEROCYCLIC DERIVATIVES AS PPAR MODULATORS ELI LILLY AND COMPANY (US) 2004-07-29 WO disclosed