SCHEMBL5597459

SCHEMBL5597459

COc1ccc(-c2cnc3nc(N)nc(N4CCNCC4C(=O)Nc4ccccc4C)c3n2)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 6/20 0.51
STK17B O94768 2/20 0.41
STK17A Q9UEE5 1/20 0.41
CHEK1 O14757 2/20 0.40
NEK2 P51955 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
DHODH Q02127 1/20 0.37
AMY1A P0DUB6 1/20 0.36
MAP3K11 Q16584 1/20 0.36
GAK O14976 1/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
ATR Q13535 1/20 0.36
MAP4K1 Q92918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5457330 0.91 NOS1 (0.53) NOS1STK17BSTK17ACHEK1NEK2
SCHEMBL5463628 0.88 NOS1 (0.51) NOS1STK17BSTK17ANEK2PDE4A
SCHEMBL5470249 0.86 NOS1 (0.51) NOS1STK17BNEK2DHODH
SCHEMBL5463636 0.86 NOS1 (0.51) NOS1STK17BSTK17ACHEK1NEK2
SCHEMBL6064705 0.86 NOS1 (0.60) NOS1STK17BSTK17ANEK2PDE4A
SCHEMBL5461836 0.85 NOS1 (0.51) NOS1STK17BSTK17ANEK2PDE4A
SCHEMBL5466005 0.84 NOS1 (0.54) NOS1STK17BSTK17ACHEK1NEK2
SCHEMBL5464734 0.84 NOS1 (0.57) NOS1STK17BSTK17ANEK2PDE4A
SCHEMBL5469822 0.84 NOS1 (0.62) NOS1STK17BSTK17ANEK2PDE4A
SCHEMBL5461552 0.83 NOS1 (0.53) NOS1STK17BSTK17ACHEK1NEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673092-B1 HETEROCYCLE-SUBSTITUTED PTERIDINE DERIVATIVES AND THEIR USE IN THERAPY 4 AZA IP NV (BE) 2007-08-15 EP disclosed