SCHEMBL5598387

SCHEMBL5598387

CCc1nc2cc(C(N)=O)ccc2n1CC

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.72
JAK2 O60674 10/20 0.60
JAK1 P23458 10/20 0.60
TYK2 P29597 10/20 0.60
JAK3 P52333 10/20 0.60
KDM4E B2RXH2 3/20 0.51
HDAC6 Q9UBN7 1/20 0.51
THRB P10828 3/20 0.50
PTGER4 P35408 2/20 0.50
MEN1 O00255 2/20 0.50
ALDH1A1 P00352 2/20 0.50
S1PR1 P21453 1/20 0.50
FGB P02675 1/20 0.50
POLB P06746 1/20 0.50
RECQL P46063 1/20 0.50
MAPT P10636 2/20 0.49
NPC1 O15118 1/20 0.49
NLRP3 Q96P20 1/20 0.49
HSP90AA1 P07900 1/20 0.48
HSP90AB1 P08238 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24688431 0.87 KMT2A (0.61) KMT2AKDM4EHDAC6THRBPTGER4
SCHEMBL18191353 0.84 KMT2A (1.00) KMT2AJAK2JAK1TYK2JAK3
SCHEMBL19437503 0.84 KMT2A (0.74) KMT2AJAK2JAK1TYK2JAK3
SCHEMBL24688398 0.83 KDM4E (0.74) KMT2AKDM4EHDAC6PTGER4MEN1
SCHEMBL22533357 0.81 KMT2A (0.52) KMT2AJAK2JAK1TYK2JAK3
SCHEMBL27442475 0.80 KMT2A (0.51) KMT2AJAK2JAK1TYK2JAK3
SCHEMBL6445182 0.79 HSD17B10 (0.59) KMT2AJAK2JAK1TYK2JAK3
SCHEMBL6445163 0.79 JAK2 (0.76) KMT2AJAK2JAK1TYK2JAK3
SCHEMBL19437515 0.76 KMT2A (0.63) KMT2AJAK2JAK1TYK2JAK3
SCHEMBL13677356 0.75 NLRP3 (0.60) KMT2AKDM4EMEN1ALDH1A1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007091950-A1 BENZIMIDAZOLES AND IMIDAZOPYRIDINES USEFUL IN THE TREATMENT OF DISEASES OR DISORDERS ASSOCIATED WITH CANNABINOID RECEPTOR 2 (CB2) SUCH AS PAIN ASTRAZENECA AB (SE) 2007-08-16 WO disclosed