SCHEMBL5599526

SCHEMBL5599526

CC1(C)CC(c2ccc(-c3ccc(CO)cc3)cc2)CC(C)(C)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.36
ATP1A1 P05023 2/20 0.35
ATP1B1 P05026 2/20 0.35
ATP1A3 P13637 2/20 0.35
ATP1B2 P14415 2/20 0.35
ATP1A2 P50993 2/20 0.35
ATP1B3 P54709 2/20 0.35
FXYD2 P54710 2/20 0.35
ATP1A4 Q13733 2/20 0.35
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
PTGS2 P35354 1/20 0.33
ADAMTS4 O75173 1/20 0.32
KIF11 P52732 1/20 0.32
HDAC2 Q92769 1/20 0.31
ESR2 Q92731 4/20 0.31
ESR1 P03372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6508796 0.95 ATP1A1 (0.37) KDM1AATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL5599819 0.85 PRKCI (0.45) ADAMTS4
SCHEMBL5787848 0.78 MAP4K1 (0.39) KDM1APDK2PDCD1CD274
SCHEMBL3138855 0.74 ESR2 (0.53) ESR2ESR1CYP3A4CYP2C9
SCHEMBL7143570 0.73
SCHEMBL14048316 0.72 ESR2 (0.56) KDM1AMKNK1MKNK2ESR2ESR1
SCHEMBL14538178 0.72 NOTUM (0.44) ESR2ESR1CYP3A4CYP2D6CYP2C9
SCHEMBL742590 0.69 ESR2 (0.52) ESR2ESR1CYP3A4CYP2D6CYP2C9
SCHEMBL6139569 0.69 L3MBTL1 (0.39)
SCHEMBL5790382 0.69 MAPT (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007500705-A 2007-01-18 JP claimed
EP-1667955-A2 CYCLOALKYLIDENE COMPOUNDS AS MODULATORS OF THE ESTROGEN RECEPTOR SmithKline Beecham Corporation (US) 2006-06-14 EP claimed
WO-2005012220-A2 CYCLOALKYLIDENE COMPOUNDS AS MODULATORS OF ESTROGEN RECEPTOR SMITHKLINE BEECHAM CORPORATION (US) 2005-02-10 WO claimed
EP-1667955-A2 CYCLOALKYLIDENE COMPOUNDS AS MODULATORS OF THE ESTROGEN RECEPTOR SmithKline Beecham Corporation (US) 2006-06-14 EP disclosed
WO-2005012220-A9 CYCLOALKYLIDENE COMPOUNDS AS MODULATORS OF ESTROGEN RECEPTOR SMITHKLINE BEECHAM CORP (US) 2005-05-19 WO disclosed
WO-2005012220-A2 CYCLOALKYLIDENE COMPOUNDS AS MODULATORS OF ESTROGEN RECEPTOR SMITHKLINE BEECHAM CORPORATION (US) 2005-02-10 WO disclosed