SCHEMBL5599568

SCHEMBL5599568

Cn1ccnc1C(CO)c1ccccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
CYP2D6 P10635 1/20 0.45
MAPT P10636 1/20 0.42
FFAR1 O14842 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KDM5A P29375 1/20 0.40
KMT2A Q03164 4/20 0.40
TDP1 Q9NUW8 1/20 0.40
PGR P06401 1/20 0.39
MEN1 O00255 1/20 0.38
CYP19A1 P11511 1/20 0.37
CNR1 P21554 1/20 0.37
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599443 0.76 KDM4E (0.46) KDM4ECYP2D6MAPTFFAR1L3MBTL1
SCHEMBL5441988 0.75 KDM4E (0.40) KDM4ECYP2D6MAPTFFAR1L3MBTL1
SCHEMBL5615786 0.74 KDM4E (0.41) KDM4ECYP2D6MAPTFFAR1L3MBTL1
SCHEMBL5599337 0.71 KDM4E (0.49) KDM4ECYP2D6MAPTFFAR1L3MBTL1
SCHEMBL9379077 0.70 CYP2D6 (0.46) KDM4ECYP2D6MAPTL3MBTL1KDM5A
SCHEMBL1503496 0.69 KDM4E (0.63) KDM4ECYP2D6MAPTFFAR1L3MBTL1
SCHEMBL10879078 0.69 CYP2D6 (0.42) CYP2D6KMT2AKCNH2
SCHEMBL5600881 0.69 FFAR1 (0.53) KDM4ECYP2D6MAPTFFAR1L3MBTL1
SCHEMBL4057807 0.69 KDM4E (0.52) KDM4ECYP2D6MAPTL3MBTL1KMT2A
SCHEMBL15358494 0.68 KDM4E (0.61) KDM4ECYP2D6MAPTL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1755678-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-02-28 EP disclosed
WO-2005097192-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-10-20 WO disclosed