SCHEMBL5599337

SCHEMBL5599337

Cn1ccnc1C(CO)c1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.46
MAPT P10636 1/20 0.44
FFAR1 O14842 8/20 0.43
CYP19A1 P11511 2/20 0.42
KMT2A Q03164 1/20 0.41
CYP2D6 P10635 1/20 0.40
RPS6KB1 P23443 1/20 0.38
LDHA P00338 1/20 0.37
LDHB P07195 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599142 0.84 FFAR1 (0.52) KDM4EL3MBTL1MAPTFFAR1KMT2A
SCHEMBL5600881 0.82 FFAR1 (0.53) KDM4EL3MBTL1MAPTFFAR1CYP2D6
SCHEMBL4899087 0.80 KDM4E (0.71) KDM4EL3MBTL1MAPTCYP19A1KMT2A
SCHEMBL5599443 0.78 KDM4E (0.46) KDM4EL3MBTL1MAPTFFAR1CYP2D6
SCHEMBL1396167 0.76 KDM4E (0.45) KDM4EL3MBTL1MAPTFFAR1CYP19A1
SCHEMBL10611537 0.73 SLC1A2 (0.44) CYP19A1KMT2A
SCHEMBL11670360 0.72 L3MBTL1 (0.67) KDM4EL3MBTL1MAPTFFAR1KMT2A
SCHEMBL6980610 0.72 TRPA1 (0.43) CYP19A1
SCHEMBL5599264 0.71 KDM4E (0.41) KDM4EL3MBTL1MAPTFFAR1KMT2A
SCHEMBL1503496 0.71 KDM4E (0.63) KDM4EL3MBTL1MAPTFFAR1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1746986-A1 ACTIVE SUBSTANCE COMBINATION COMPRISING A CARBINOL COMBINED TO AT LEAST AN NSAID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-01-31 EP claimed
WO-2005097099-A1 ACTIVE SUBSTANCE COMBINATION COMPRISING A CARBINOL COMBINED TO AT LEAST AN NSAID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-10-20 WO claimed
EP-1755678-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-02-28 EP disclosed
WO-2005097192-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-10-20 WO disclosed