SCHEMBL560042

SCHEMBL560042

COC(=O)CSCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.59
FFAR1 O14842 1/20 0.59
HTT P42858 2/20 0.57
GAA P10253 1/20 0.57
L3MBTL1 Q9Y468 2/20 0.55
RAB9A P51151 5/20 0.54
CYP1A2 P05177 2/20 0.53
CYP2C19 P33261 2/20 0.52
LMNA P02545 1/20 0.51
ALDH1A1 P00352 4/20 0.50
NPC1 O15118 2/20 0.50
HPGD P15428 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
PKM P14618 2/20 0.49
ALOX15 P16050 2/20 0.49
HSD17B10 Q99714 2/20 0.49
RXFP1 Q9HBX9 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11464189 0.90 ACE (0.51) MAPK1FFAR1HTTGAAL3MBTL1
SCHEMBL15745228 0.86 NPC1 (0.56) FFAR1RAB9ALMNAALDH1A1NPC1
SCHEMBL8895881 0.84 CYP2C19 (0.66) MAPK1FFAR1HTTGAARAB9A
SCHEMBL13870189 0.83 MAPT (0.58) L3MBTL1RAB9ACYP1A2CYP2C19ALDH1A1
Acetic Acid Methyl Ester SCHEMBL23070551 0.82 CYP2C19 (0.53) MAPK1FFAR1HTTGAAL3MBTL1
SCHEMBL5410393 0.81 GAA (0.61) HTTGAARAB9ACYP1A2LMNA
SCHEMBL10953947 0.81 ALDH1A1 (0.46) MAPK1FFAR1HTTGAACYP1A2
SCHEMBL3256326 0.81 NPC1 (0.62) HTTGAAL3MBTL1RAB9ACYP2C19
SCHEMBL11265645 0.81 ALDH1A1 (0.61) MAPK1GAARAB9ACYP1A2CYP2C19
SCHEMBL9069764 0.81 CYP2C19 (0.57) MAPK1FFAR1HTTGAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116478132-A 2, 5-disubstituted and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-07-25 CN disclosed
CN-116478131-A 2, 5-disubstituted and 2,5, 6-trisubstituted 3-methylpyrazines as allosteric SHP2 inhibitors 锐新医药公司 2023-07-25 CN disclosed
CN-110523541-B Alkyl thioether ether ethyl hydroximic acid medicament and preparation method and application thereof 中南大学 2021-09-28 CN disclosed
US-20210276023-A1 ALKYL THIOETHER ETHYL HYDROXAMIC ACID BENEFICIATION REAGENT AND PREPARATION METHOD AND APPLICATION THEREOF CENTRAL SOUTH UNIVERSITY (CN) 2021-09-09 US disclosed
CN-106588720-B Sulfidomethyl amphyl preparation method and application based on dual catalyst system 中国科学院宁波材料技术与工程研究所 2019-06-11 CN disclosed
CN-106588720-A Dual catalytic system based sulfur methyl phenol derivative preparation method and application 中国科学院宁波材料技术与工程研究所 2017-04-26 CN disclosed
EP-1849796-B1 ANTI-PENICILLIN RESISTANT PNEUMOCOCCI AGENT AND NOVEL 16-MEMBERED RING MACROLIDE DERIVATIVE MICROBIAL CHEM RES FOUND (JP) 2014-11-05 EP disclosed
US-8507453-B2 Anti-penicillin resistant pneumococci agent and novel 16-membered macrolide derivative MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 2013-08-13 US disclosed
US-8507453-B2 Anti-penicillin resistant pneumococci agent and novel 16-membered macrolide derivative MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 2013-08-13 US disclosed
US-8420698-B2 Histone deacetylase inhibitors ERRANT GENE THERAPEUTICS, LLC (US) 2013-04-16 US disclosed
EP-1408946-A4 HISTONE DEACETYLASE INHIBITORS CIRCAGEN PHARMACEUTICAL (US) 2004-06-09 EP disclosed
EP-1408946-A2 HISTONE DEACETYLASE INHIBITORS Circagen Pharmaceutical (US) 2004-04-21 EP disclosed
US-20030125306-A1 Histone deacetylase inhibitors CIRCAGEN PHARMACEUTICAL, A DELAWARE CORPORATION 2003-07-03 US disclosed
US-20030083521-A1 Such as 5-phenyl-2,4-pentadienoylhydroxamic acid; for treating cancer, hematopoiesis, and genetic metabolic disorders (cystic fibrosis and adrenoleukodystrophy) CIRCAGEN PHARMACEUTICAL, A MARYLAND CORPORATION 2003-05-01 US disclosed
US-6495719-B2 FOR USE IN THERAPY OF CANCER, HEMATOLOGICAL DISORDERS, SUCH AS HEMATOPOIESIS, AND GENETIC RELATED METABOLIC DISORDERS, SUCH AS, CYSTIC FIBROSIS AND ADRENOLEUKODYSTROPHY CIRCAGEN PHARMACEUTICAL 2002-12-17 US disclosed
US-20020143196-A1 Histone deacetylase inhibitors ERRANT GENE THERAPEUTICS, LLC 2002-10-03 US disclosed
US-20020143052-A1 Histone deacetylase inhibitors ANGELA CHEN SABELLA 2002-10-03 US disclosed
WO-2002076941-A2 HISTONE DEACETYLASE INHIBITORS CIRCAGEN PHARMACEUTICAL (US) 2002-10-03 WO disclosed
US-20020143037-A1 Histone deacetylase inhibitors CIRCAGEN PHARMACEUTICAL, A DELAWARE CORPORATION 2002-10-03 US disclosed
US-3988375-A HERBICIDES MONSANTO COMPANY (US) 1976-10-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030083521-A1 Such as 5-phenyl-2,4-pentadienoylhydroxamic acid; for treating cancer, hematopoiesis, and genetic metabolic disorders (cystic fibrosis and adrenoleukodystrophy) ZFX, HDAC5, ZNF277 MAPK1 3331/4885FFAR1 1640/4885HTT 2997/4885
US-20020143052-A1 Histone deacetylase inhibitors HDAC1, HDAC11, HDAC9 MAPK1 3264/4885FFAR1 3522/4885HTT 1868/4885
US-20030125306-A1 Histone deacetylase inhibitors HDAC1, HDAC11, HDAC9 MAPK1 3264/4885FFAR1 3522/4885HTT 1868/4885
US-20020143196-A1 Histone deacetylase inhibitors HDAC1, HDAC11, HDAC5 MAPK1 3260/4885FFAR1 3679/4885HTT 2627/4885
US-20020143037-A1 Histone deacetylase inhibitors HDAC1, HDAC9, HDAC11 MAPK1 3365/4885FFAR1 3282/4885HTT 2627/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.