SCHEMBL5605847

SCHEMBL5605847

CN(C)C1Cc2cc(-c3ccccc3)cc(-c3ccccc3Cl)c2O1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.39
HTR7 P34969 7/20 0.39
SLC6A9 P48067 4/20 0.38
CYP2A6 P11509 1/20 0.36
AQP1 P29972 3/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
HTR2A P28223 2/20 0.31
HTR2C P28335 2/20 0.31
HTR2B P41595 2/20 0.31
HRH3 Q9Y5N1 2/20 0.31
HSD11B1 P28845 1/20 0.31
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5605603 0.84 HTR1A (0.44) HTR1AHTR7SLC6A9PTGS1PTGS2
SCHEMBL5583714 0.83 CNR1 (0.39) HTR1AHTR7SLC6A9CYP2A6AQP1
SCHEMBL5605796 0.81 MAPK14 (0.40) HTR1AHTR7
SCHEMBL5583710 0.81 CYP2A6 (0.39) HTR1AHTR7SLC6A9CYP2A6AQP1
SCHEMBL5605843 0.78 CNR1 (0.34) HTR1AHTR7SLC6A9CYP2A6AQP1
SCHEMBL4220714 0.78 AQP1 (0.54) SLC6A9CYP2A6AQP1HRH3
SCHEMBL4230563 0.77 AQP1 (0.57) SLC6A9CYP2A6AQP1HRH3
SCHEMBL4230569 0.76 AQP1 (0.44) SLC6A9CYP2A6AQP1HRH3
SCHEMBL4596667 0.73 AQP1 (0.43) HTR1AHTR7SLC6A9AQP1
SCHEMBL15758987 0.72 AKR1C2 (0.37) SLC6A9HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007509174-A 2007-04-12 JP claimed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP claimed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO claimed