SCHEMBL5606006

SCHEMBL5606006

COC(=O)c1ccc2cc(-c3ccc(OC)cc3)ccc2c1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.65
CA2 P00918 1/20 0.65
PLAU P00749 9/20 0.62
PLAT P00750 4/20 0.62
PLG P00747 2/20 0.62
CYP11B1 P15538 2/20 0.61
CYP11B2 P19099 2/20 0.61
CYP19A1 P11511 1/20 0.61
KMT2A Q03164 2/20 0.55
KDM4E B2RXH2 2/20 0.53
MEN1 O00255 1/20 0.53
MAPT P10636 1/20 0.53
PTPN11 Q06124 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30698055 1.00 CA1 (0.65) CA1CA2PLAUPLATPLG
SCHEMBL13900228 0.91 CYP11B1 (0.69) CA1CA2PLAUPLATPLG
SCHEMBL15897010 0.90 CYP11B1 (0.69) CA1CA2PLAUPLATPLG
SCHEMBL2112531 0.87 CA12 (0.61) CA1CA2PLAUPLATPLG
SCHEMBL2311608 0.87 CYP19A1 (0.69) CA1CA2PLAUPLATPLG
SCHEMBL1856468 0.86 KDM4E (0.70) CA1CA2PLAUPLATPLG
SCHEMBL16604876 0.86 CA1 (0.88) CA1CA2KMT2AKDM4EMEN1
SCHEMBL269558 0.86 CA1 (0.88) CA1CA2KMT2AKDM4EMEN1
SCHEMBL5224416 0.85 APP (0.56) CA1CA2PLAUPLATPLG
SCHEMBL13486839 0.85 CYP1A2 (0.60) CA1CA2PLAUPLATPLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117700298-A Preparation method of hydroxyl adapalene 湖北广济药业股份有限公司 2024-03-15 CN claimed
CN-111333496-B Preparation method of adapalene 武汉诺安药业有限公司 2023-10-13 CN claimed
EP-0358574-B1 PROCESS FOR THE PREPARATION OF ADAMANTANE-1 DERIVATIVES CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA - CIRD GALDERMA (FR) 1993-02-17 EP claimed
CN-117700298-A Preparation method of hydroxyl adapalene 湖北广济药业股份有限公司 2024-03-15 CN disclosed
CN-117700298-A Preparation method of hydroxyl adapalene 湖北广济药业股份有限公司 2024-03-15 CN disclosed
CN-111333496-B Preparation method of adapalene 武汉诺安药业有限公司 2023-10-13 CN disclosed
CN-111333496-B Preparation method of adapalene 武汉诺安药业有限公司 2023-10-13 CN disclosed
CN-111333496-A Preparation method of adapalene 武汉诺安药业有限公司 2020-06-26 CN disclosed
WO-2007125542-A2 A PROCESS FOR PREPARATION OF ADAPALENE USV LIMITED (IN) 2007-11-08 WO disclosed
US-5015758-A Process for the preparation of 1-adamantane derivatives CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (CIRD) (FR) 1991-05-14 US disclosed