SCHEMBL5608528

SCHEMBL5608528

CCCCN(CCCC)c1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
KCNA5 P22460 2/20 0.48
KCNN4 O15554 1/20 0.48
TRPV1 Q8NER1 1/20 0.46
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
S1PR1 P21453 1/20 0.42
CHRNB2 P17787 3/20 0.41
CHRNA4 P43681 3/20 0.41
CHRNA7 P36544 1/20 0.41
HTT P42858 1/20 0.40
LMNA P02545 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18929879 0.93 L3MBTL1 (0.46) L3MBTL1TDP1KCNA5KCNN4TRPV1
SCHEMBL10771297 0.84 TRPV1 (0.48) L3MBTL1TDP1KCNA5KCNN4TRPV1
SCHEMBL27463798 0.81 KCNA5 (0.51) L3MBTL1TDP1KCNA5KCNN4TRPV1
SCHEMBL17484099 0.81 KCNA5 (0.48) L3MBTL1TDP1KCNA5KCNN4TRPV1
SCHEMBL1432726 0.80 NPSR1 (0.51) L3MBTL1KCNA5KCNN4CYP3A4CYP2C19
SCHEMBL17059858 0.78 KCNA5 (0.46) L3MBTL1TDP1KCNA5KCNN4TRPV1
SCHEMBL11490914 0.77 L3MBTL1 (0.49) L3MBTL1TDP1KCNA5KCNN4TRPV1
SCHEMBL811561 0.76 NR1H2 (0.50) CYP3A4CYP2D6HTTMAPTMAPK1
SCHEMBL107013 0.76 CNR2 (0.49) TDP1LMNAPOLBMAPTNPSR1
SCHEMBL14229682 0.75 TP53 (0.56) L3MBTL1KCNA5KCNN4TRPV1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed
EP-1354887-A1 Ligands for metals and improved metal-catalyzed processes based thereon Massachusetts Insitute of Technology (US) 2003-10-22 EP disclosed