SCHEMBL5608566

SCHEMBL5608566

CCS(=O)(=O)c1ccc(-c2cc(C(F)F)nn2-c2ccc(S(N)(=O)=O)cc2)cc1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.79
PTGS1 P23219 12/20 0.79
ABCB11 O95342 2/20 0.66
ALDH1A1 P00352 1/20 0.66
CHRNA7 P36544 1/20 0.54
PDPK1 O15530 2/20 0.54
CA1 P00915 2/20 0.54
CA2 P00918 2/20 0.54
CA9 Q16790 2/20 0.54
PTGES O14684 1/20 0.54
HDAC3 O15379 1/20 0.54
CA12 O43570 1/20 0.54
PDE5A O76074 1/20 0.54
MT-CO2 P00403 1/20 0.54
LMNA P02545 1/20 0.54
CA3 P07451 1/20 0.54
CYP3A4 P08684 1/20 0.54
ALOX5 P09917 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
CYP2D6 P10635 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL213150 0.88 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL3243184 0.88 PTGS2 (0.82) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6352647 0.87 PTGS2 (0.80) PTGS2PTGS1ABCB11ALDH1A1CHRNA7
SCHEMBL27435791 0.86 PTGS2 (0.75) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL3249718 0.86 PTGS2 (0.95) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL7789562 0.86 PTGS2 (0.78) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL212658 0.86 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1CHRNA7
SCHEMBL6339240 0.86 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1CHRNA7
SCHEMBL215341 0.85 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL6339195 0.85 PTGS2 (0.90) PTGS2PTGS1ABCB11ALDH1A1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1039914-A4 CYCLOOXYGENASE-2 INHIBITION CORNELL RES FOUNDATION INC (US) 2007-06-27 EP disclosed
EP-1039914-A1 CYCLOOXYGENASE-2 INHIBITION CORNELL RESEARCH FOUNDATION, INC. (US) 2000-10-04 EP disclosed
WO-1999030721-A1 CYCLOOXYGENASE-2 INHIBITION CORNELL RESEARCH FOUNDATION, INC. (US) 1999-06-24 WO disclosed