SCHEMBL5608680

SCHEMBL5608680

Cc1ccc(C)c(NC2CC2)c1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
KDM4E B2RXH2 3/20 0.54
POLB P06746 1/20 0.54
RAPGEF4 Q8WZA2 2/20 0.52
HDAC8 Q9BY41 1/20 0.47
GAA P10253 3/20 0.44
HTT P42858 2/20 0.42
TP53 P04637 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
P2RX7 Q99572 1/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5608474 0.90 HDAC8 (0.59) ALDH1A1KDM4EPOLBRAPGEF4HDAC8
SCHEMBL82947 0.87 BRD4 (0.48) ALDH1A1KDM4EPOLBRAPGEF4HDAC8
Hydrochloric Acid SCHEMBL69124 0.86 BRD4 (0.47) ALDH1A1KDM4EPOLBRAPGEF4HDAC8
SCHEMBL12327879 0.82 GLA (0.48) ALDH1A1KDM4EPOLBRAPGEF4GAA
SCHEMBL30657543 0.80 KDM4E (0.46) ALDH1A1KDM4EPOLBRAPGEF4GAA
SCHEMBL20345722 0.80 KDM4E (0.46) ALDH1A1KDM4EPOLBRAPGEF4GAA
SCHEMBL28791583 0.79 MEN1 (0.48) HDAC8GAATP53
SCHEMBL2637117 0.78 MEN1 (0.47) HDAC8GAATP53
SCHEMBL30777245 0.77 P2RX7 (0.44) ALDH1A1KDM4EPOLBHDAC8GAA
SCHEMBL16418620 0.77 HDAC8 (0.43) ALDH1A1KDM4EPOLBHDAC8HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed
EP-1354887-A1 Ligands for metals and improved metal-catalyzed processes based thereon Massachusetts Insitute of Technology (US) 2003-10-22 EP disclosed
EP-1097158-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-05-09 EP disclosed
WO-2000002887-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-01-20 WO disclosed