SCHEMBL5608474

SCHEMBL5608474

Cc1ccc(C)c(NC2CCCCC2)c1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.59
ALDH1A1 P00352 4/20 0.58
KDM4E B2RXH2 4/20 0.58
POLB P06746 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.51
RAPGEF4 Q8WZA2 1/20 0.47
LMNA P02545 3/20 0.46
MAPT P10636 2/20 0.46
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
GAA P10253 3/20 0.45
TP53 P04637 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ADRB2 P07550 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5608680 0.90 ALDH1A1 (0.54) HDAC8ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL13801923 0.84 HDAC8 (0.57) HDAC8ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL82947 0.82 BRD4 (0.48) HDAC8ALDH1A1KDM4EPOLBRAPGEF4
SCHEMBL2361893 0.82 KDM4E (0.59) HDAC8ALDH1A1KDM4EPOLBL3MBTL1
Hydrochloric Acid SCHEMBL69124 0.81 BRD4 (0.47) HDAC8ALDH1A1KDM4EPOLBRAPGEF4
SCHEMBL1341748 0.80 KDM4E (0.56) HDAC8ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL13663589 0.80 HDAC8 (0.54) HDAC8ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL11847765 0.80 ALDH1A1 (0.46) HDAC8ALDH1A1KDM4EL3MBTL1LMNA
SCHEMBL3674808 0.79 NPC1 (0.51) HDAC8ALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL18010743 0.79 ALDH1A1 (0.49) HDAC8ALDH1A1KDM4EPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed
EP-1354887-A1 Ligands for metals and improved metal-catalyzed processes based thereon Massachusetts Insitute of Technology (US) 2003-10-22 EP disclosed
EP-1097158-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-05-09 EP disclosed
WO-2000002887-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-01-20 WO disclosed