SCHEMBL5617569

SCHEMBL5617569

C=CCc1ccc(-c2ccccc2)c(P)c1CC=C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.36
GABRB2 P47870 2/20 0.36
AURKA O14965 1/20 0.32
DAPK3 O43293 1/20 0.32
MAP4K4 O95819 1/20 0.32
RET P07949 1/20 0.32
IGF1R P08069 1/20 0.32
MET P08581 1/20 0.32
PIM1 P11309 1/20 0.32
LTK P29376 1/20 0.32
KDR P35968 1/20 0.32
MAPK8 P45983 1/20 0.32
MAPK9 P45984 1/20 0.32
CDK8 P49336 1/20 0.32
CLK2 P49760 1/20 0.32
CDK9 P50750 1/20 0.32
CDK5 Q00535 1/20 0.32
ACVR1 Q04771 1/20 0.32
PTK2 Q05397 1/20 0.32
MAP4K2 Q12851 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5403133 0.86 GABRA1 (0.40) GABRA1GABRB2AURKADAPK3MAP4K4
SCHEMBL9859732 0.81 GABRA1 (0.37) GABRA1GABRB2AURKADAPK3MAP4K4
SCHEMBL8605193 0.80 GABRA1 (0.36) GABRA1GABRB2AURKADAPK3MAP4K4
SCHEMBL1646863 0.80 GABRA1 (0.36) GABRA1GABRB2AURKADAPK3MAP4K4
SCHEMBL2362467 0.77 GABRA1 (0.52) GABRA1GABRB2AURKADAPK3MAP4K4
SCHEMBL9504989 0.77 GABRA1 (0.36) GABRA1GABRB2AURKADAPK3MAP4K4
SCHEMBL10766912 0.76 ALDH1A1 (0.38) GABRA1GABRB2KMT2AMEN1MAPT
Bromide SCHEMBL27823869 0.75 GABRA1 (0.49) GABRA1GABRB2AURKADAPK3MAP4K4
SCHEMBL27886719 0.74 GABRA1 (0.47) GABRA1GABRB2AURKADAPK3MAP4K4
SCHEMBL2362270 0.74 GABRA1 (0.39) GABRA1GABRB2AURKADAPK3MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1354887-B1 Ligands for metals and improved metal-catalyzed processes based thereon MASSACHUSETTS INST TECHNOLOGY (US) 2007-04-25 EP disclosed
EP-1097158-B1 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INST TECHNOLOGY (US) 2006-01-25 EP disclosed
EP-1354887-A1 Ligands for metals and improved metal-catalyzed processes based thereon Massachusetts Insitute of Technology (US) 2003-10-22 EP disclosed
EP-1097158-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2001-05-09 EP disclosed
WO-2000002887-A2 LIGANDS FOR METALS AND METAL-CATALYZED PROCESSES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-01-20 WO disclosed