SCHEMBL5617833

SCHEMBL5617833

CCOc1ccc(C(O)c2ccnn2C)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.58
LMNA P02545 2/20 0.50
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
TAS1R2 Q8TE23 1/20 0.44
ALDH1A1 P00352 4/20 0.44
MAPT P10636 2/20 0.43
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NQO1 P15559 1/20 0.41
LTA4H P09960 3/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4910223 0.83 ALDH1A1 (0.50) L3MBTL1ALDH1A1MAPTRAB9ACYP1A2
SCHEMBL4908140 0.78 CYP3A4 (0.42) LMNAALDH1A1SMN1; SMN2CYP3A4CYP2D6
SCHEMBL7589137 0.77 KDM4E (0.50) LMNAALDH1A1SMN1; SMN2CYP19A1KDM4E
SCHEMBL7590836 0.77 KDM4E (0.50) LMNAALDH1A1SMN1; SMN2CYP19A1KDM4E
SCHEMBL2788882 0.77 KDM4E (0.50) LMNAALDH1A1SMN1; SMN2CYP19A1KDM4E
SCHEMBL9114461 0.77 NQO1 (0.64) L3MBTL1LMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL31040269 0.76 SMN1; SMN2 (0.41) L3MBTL1LMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL6920072 0.76 MAPK1 (0.45) LMNASMN1; SMN2CYP1A2CYP19A1KDM4E
SCHEMBL4899497 0.76 HTT (0.45) LMNAALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL17865259 0.76 CYP3A4 (0.42) LMNAMAPTSMN1; SMN2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1755678-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-02-28 EP disclosed
WO-2005097192-A2 ACTIVE SUBSTANCE COMBINATION OF A CARBINOL COMPOUND AND AN OPIOID LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2005-10-20 WO disclosed