SCHEMBL5618062

SCHEMBL5618062

O=Cc1ccc2c(ccc3ccccc32)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
HSD17B10 Q99714 2/20 0.54
CYP1B1 Q16678 2/20 0.54
HIF1A Q16665 2/20 0.54
HPRT1 P00492 4/20 0.52
KIF11 P52732 2/20 0.52
CYP2A6 P11509 1/20 0.50
TSHR P16473 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
HPGD P15428 2/20 0.47
MAPT P10636 1/20 0.47
ERN1 O75460 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CYP1A2 P05177 3/20 0.44
ERBB2 P04626 1/20 0.44
FYN P06241 1/20 0.44
MAOA P21397 1/20 0.44
ACHE P22303 1/20 0.44
AHR P35869 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29913753 1.00 ALDH1A1 (0.54) ALDH1A1HSD17B10CYP1B1HIF1AHPRT1
SCHEMBL27456577 0.98 ALDH1A1 (0.52) ALDH1A1HSD17B10CYP1B1HIF1AHPRT1
SCHEMBL10484075 0.98 HPRT1 (0.56) ALDH1A1HSD17B10CYP1B1HIF1AHPRT1
SCHEMBL11622042 0.90 AKR1B1 (0.49) ALDH1A1HSD17B10CYP1B1HIF1AHPRT1
SCHEMBL10484322 0.90 HPRT1 (0.56) ALDH1A1HSD17B10CYP1B1HIF1AHPRT1
SCHEMBL30811866 0.90 HPRT1 (0.56) ALDH1A1HSD17B10CYP1B1HIF1AHPRT1
SCHEMBL5617799 0.89 ALDH1A1 (0.56) ALDH1A1HSD17B10CYP1B1HIF1AHPRT1
SCHEMBL9127399 0.89 CYP2A6 (0.48) ALDH1A1HSD17B10KIF11CYP2A6TSHR
SCHEMBL10348677 0.88 ALDH1A1 (0.50) ALDH1A1HSD17B10CYP1B1HIF1AHPRT1
SCHEMBL9798242 0.87 CYP2A6 (0.44) ALDH1A1HSD17B10CYP1B1HIF1AKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 71 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103391945-B Isoxazolidine derivant 奇斯药制品公司 2016-11-09 CN claimed
CN-103391945-A Isoxazolidine derivatives CHIESI FARMA SPA 2013-11-13 CN claimed
CN-103380142-A Isoxazolidine derivatives CHIESI FARMA SPA 2013-10-30 CN claimed
CN-101282987-A Glucocorticoid 16alpha,17alpha-isoxazolidines as anti-inflammatory agents NOVARTIS AG (CH) 2008-10-08 CN claimed
CN-1284781-C Polycyclic compounds with antitumor activity HOFFMANN LA ROCHE (CH) 2006-11-15 CN claimed
CN-1610681-A Polycyclic compounds having anti-tumor activity HOFFMANN LA ROCHE (CH) 2005-04-27 CN claimed
CN-114956933-A Marker containing isotope oxygen atom and preparation method and application thereof 清华大学 2022-08-30 CN disclosed
CN-111517902-B Aerobic oxidation system containing sulfinic acid, sulfonic acid or derivatives thereof and photo-oxidation promoting method thereof 清华大学 2022-06-14 CN disclosed
CN-106565622-B Novel isoxazoles, process for their preparation and their use 尚科纺织企业工业及贸易公司 2022-02-15 CN disclosed
WO-2021129639-A1 ORGANIC COMPOUND AND APPLICATION, AND ORGANIC ELECTROLUMINESCENCE DEVICE USING ORGANIC COMPOUND 陕西莱特光电材料股份有限公司 2021-07-01 WO disclosed
CN-111517902-A Aerobic oxidation system containing sulfinic acid, sulfonic acid or derivatives thereof and photo-oxidation promoting method thereof 清华大学 2020-08-11 CN disclosed
WO-2020155595-A1 AEROBIC OXIDATION SYSTEM CONTAINING SULFINIC ACID, SULFONIC ACID OR DERIVATIVES THEREOF AND PHOTOCATALYTIC OXIDATION METHOD THEREFOR 清华大学 2020-08-06 WO disclosed
CN-110386926-A A kind of organic photoelectrical material and its preparation method and application containing benzheterocycle structure 武汉尚赛光电科技有限公司 2019-10-29 CN disclosed
US-4623661-A HYDROXAMIC ACID DERIVATIVES ABBOTT LABORATORIES (US) 1986-11-18 US disclosed
EP-0199151-A2 Lipoxygenase inhibiting compounds ABBOTT LABORATORIES (US) 1986-10-29 EP disclosed
EP-0172427-A2 Process for production of vinyl chloride polymer Shin-Etsu Chemical Co., Ltd. (JP) 1986-02-26 EP disclosed
US-4511582-A 2-METHYL-2-/PHENANTHRYLMETHYL/AMINOPROPANEDIOL OR ESTERS BURROUGHS WELLCOME CO. (US) 1985-04-16 US disclosed
EP-0125701-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP disclosed
US-4060677-A Process for molecular weight lowering of vinyl halide polymers employing saturated carbon to carbon bonded aldehydes HOOKER CHEMICALS & PLASTICS CORPORATION (US) 1977-11-29 US disclosed
US-3987116-A ETHYNYLARYL COMPOUNDS AND DERIVATIVES THEREOF WILLIAM H. RORER, INC. (US) 1976-10-19 US disclosed