SCHEMBL5618486

SCHEMBL5618486

Brc1cccc(CCCC2CCNC2)c1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.42
HRH3 Q9Y5N1 2/20 0.41
EP300 Q09472 1/20 0.39
GBA1 P04062 1/20 0.38
SLC6A4 P31645 1/20 0.37
PARP1 P09874 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRM3 P20309 1/20 0.36
CHRNA4 P43681 1/20 0.36
EED O75530 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17791449 0.83 MAOA (0.44) HRH3GBA1SLC6A4PARP1CHRM2
SCHEMBL12735989 0.82 TAAR1 (0.47) TAAR1HRH3EP300GBA1SLC6A4
SCHEMBL29890848 0.82 EED (0.52) TAAR1HRH3EP300GBA1SLC6A4
SCHEMBL26187550 0.82 EED (0.52) TAAR1HRH3EP300GBA1SLC6A4
SCHEMBL29889395 0.82 EED (0.52) TAAR1HRH3EP300GBA1SLC6A4
Hydrochloric Acid SCHEMBL30648851 0.81 EED (0.51) TAAR1HRH3EP300GBA1SLC6A4
SCHEMBL19524560 0.75 TAAR1 (0.46) TAAR1
Hydrochloric Acid SCHEMBL2634704 0.74 GBA1 (0.61) TAAR1EP300GBA1SLC6A4EED
SCHEMBL15130164 0.74 HRH3 (0.48) HRH3GBA1SLC6A4PARP1CHRM2
SCHEMBL11636313 0.74 SLC6A4 (0.45) HRH3GBA1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007056075-A2 SIX MEMBERED HETEROAROMATIC INHIBITORS TARGETING RESISTANT KINASE MUTATIONS TARGEGEN, INC. (US) 2007-05-18 WO disclosed