SCHEMBL5620548

SCHEMBL5620548

NC(=O)c1cccc2c1nc(N1CCCNCC1)n2CCN1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.43
PIM1 P11309 1/20 0.42
FLT3 P36888 1/20 0.42
PIM3 Q86V86 1/20 0.42
BRSK1 Q8TDC3 1/20 0.42
AURKB Q96GD4 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
DHODH Q02127 1/20 0.41
HTR3A P46098 1/20 0.40
PARP2 Q9UGN5 1/20 0.39
PARP3 Q9Y6F1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5621867 0.99 PARP1 (0.44) PARP1PIM1FLT3PIM3BRSK1
SCHEMBL5620376 0.97 PARP1 (0.45) PARP1PIM1FLT3PIM3BRSK1
SCHEMBL5620307 0.96 PARP1 (0.46) PARP1PIM1FLT3PIM3BRSK1
SCHEMBL5620405 0.89 PARP1 (0.43) PARP1HTR3A
SCHEMBL5621901 0.89 PARP1 (0.43) PARP1PIM1PIM3HTR3A
SCHEMBL5621918 0.86 PARP1 (0.44) PARP1PIM1FLT3PARP2
SCHEMBL7037841 0.86 HTR3A (0.38) PARP1HTR3A
SCHEMBL5620467 0.85 PARP1 (0.41) PARP1HTR3A
SCHEMBL5621625 0.85 PARP1 (0.41) PARP1HTR3A
SCHEMBL7046777 0.85 HTR3A (0.39) HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39608-E1 Substituted benzimidazoles and their use as PARP inhibitors ABBOTT GMBH & CO. KG (DE) 2007-05-01 US disclosed
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed