SCHEMBL7046777

SCHEMBL7046777

NC(=O)Oc1cccc2c1nc(N1CCCNCC1)n2CCN1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 4/20 0.39
NPY1R P25929 1/20 0.36
OPRK1 P41145 6/20 0.36
OPRM1 P35372 2/20 0.36
OPRD1 P41143 2/20 0.36
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
CNR2 P34972 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7037841 0.99 HTR3A (0.38) HTR3ANPY1ROPRK1OPRM1OPRD1
SCHEMBL7041533 0.97 HTR3A (0.40) HTR3ANPY1ROPRK1OPRM1OPRD1
SCHEMBL7046613 0.96 HTR3A (0.40) HTR3ANPY1ROPRK1OPRM1OPRD1
SCHEMBL7036855 0.90 HTR3A (0.40) HTR3ACHRNB2CHRNA4
SCHEMBL7044695 0.90 HTR3A (0.40) HTR3ACHRNB2CHRNA4
SCHEMBL7045753 0.88 HTR3A (0.38) HTR3ACHRNB2CHRNA4
SCHEMBL7042010 0.87 FLT3 (0.41) HTR3ACHRNB2CHRNA4
SCHEMBL7042935 0.86 HTR3A (0.42) HTR3A
SCHEMBL7042964 0.86 HTR3A (0.42) HTR3A
SCHEMBL5621867 0.85 PARP1 (0.44) HTR3AOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed