SCHEMBL5624486

SCHEMBL5624486

Cc1cc(S(=O)(=O)O)cnc1/N=C/N(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.38
CYP2C19 P33261 3/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
HTR6 P50406 3/20 0.36
L3MBTL1 Q9Y468 3/20 0.34
LMNA P02545 2/20 0.34
GAA P10253 2/20 0.34
KDM4E B2RXH2 6/20 0.34
ALDH1A1 P00352 7/20 0.32
RAB9A P51151 4/20 0.32
NPC1 O15118 3/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
HSD17B10 Q99714 2/20 0.32
HPGD P15428 2/20 0.32
POLB P06746 1/20 0.32
TSHR P16473 1/20 0.32
ALOX15 P16050 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5624489 1.00 CYP1A2 (0.38) CYP1A2CYP2C19CYP3A4CYP2D6HTR6
Dimethylformamide SCHEMBL27878591 0.71 CHRM1 (0.38) LMNAGAAKDM4EALDH1A1HTT
SCHEMBL5623766 0.68 NOS3 (0.50) LMNAGAAKDM4EALDH1A1RAB9A
SCHEMBL313339 0.65 ALDH1A1 (0.45) CYP1A2LMNAGAAKDM4EALDH1A1
SCHEMBL19555026 0.62 KMT2A (0.40) CYP1A2CYP2C19CYP3A4CYP2D6HTR6
SCHEMBL21572724 0.62 HSD17B10 (0.37) CYP1A2CYP2C19CYP3A4CYP2D6L3MBTL1
SCHEMBL32662109 0.62 HSD17B10 (0.37) CYP1A2CYP2C19CYP3A4CYP2D6L3MBTL1
SCHEMBL1202147 0.62 KMT2A (0.40) CYP1A2CYP2C19CYP3A4CYP2D6HTR6
SCHEMBL1355119 0.62 PLAU (0.47) L3MBTL1LMNAGAAKDM4EALDH1A1
SCHEMBL14181404 0.61 CYP3A4 (0.46) CYP3A4LMNAGAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7273863-B1 Benzophenones as inhibitors of reverse transcriptase SMITHKLINE BEECHAM CORPORATION (US) 2007-09-25 US disclosed
US-7273863-B1 Benzophenones as inhibitors of reverse transcriptase SMITHKLINE BEECHAM CORPORATION (US) 2007-09-25 US disclosed
EP-1710238-A1 Benzophenones as inhibitors of reverse transcriptase GLAXO GROUP LIMITED (GB) 2006-10-11 EP disclosed
EP-1208091-B1 BENZOPHENONES AS INHIBITORS OF REVERSE TRANSCRIPTASE GLAXO GROUP LTD (GB) 2006-05-03 EP disclosed
EP-1208091-A1 BENZOPHENONES AS INHIBITORS OF REVERSE TRANSCRIPTASE GLAXO GROUP LIMITED (GB) 2002-05-29 EP disclosed
WO-2001017982-A1 BENZOPHENONES AS INHIBITORS OF REVERSE TRANSCRIPTASE GLAXO GROUP LIMITED (GB) 2001-03-15 WO disclosed