SCHEMBL5632154

SCHEMBL5632154

NS(=O)(=O)Nc1ccccn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.59
ATM Q13315 1/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
KDM4E B2RXH2 7/20 0.54
LMNA P02545 2/20 0.54
ALDH1A1 P00352 4/20 0.51
HPGD P15428 1/20 0.51
HSD17B10 Q99714 1/20 0.51
POLB P06746 1/20 0.51
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
RXFP1 Q9HBX9 2/20 0.49
NPC1 O15118 1/20 0.48
PKM P14618 1/20 0.48
RAB9A P51151 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
MAPK1 P28482 1/20 0.47
MAPK10 P53779 1/20 0.47
GFER P55789 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11666645 0.89 SMN1; SMN2 (0.50) TSHRATMSMN1; SMN2KDM4ELMNA
SCHEMBL2104486 0.79 TSHR (0.59) TSHRATMSMN1; SMN2KDM4ELMNA
SCHEMBL23308872 0.79 TSHR (0.59) TSHRATMSMN1; SMN2KDM4ELMNA
SCHEMBL27673212 0.79 TSHR (0.59) TSHRATMSMN1; SMN2KDM4ELMNA
SCHEMBL1631053 0.79 TSHR (0.65) TSHRATMSMN1; SMN2KDM4ELMNA
Hydrochloric Acid SCHEMBL20502504 0.78 TSHR (0.62) TSHRATMSMN1; SMN2KDM4ELMNA
SCHEMBL3374110 0.78 KDM4E (0.62) TSHRATMSMN1; SMN2KDM4ELMNA
SCHEMBL6320584 0.76 KDM4E (0.61) TSHRATMSMN1; SMN2KDM4ELMNA
SCHEMBL30746463 0.76 TSHR (0.61) TSHRATMSMN1; SMN2KDM4ELMNA
SCHEMBL1667129 0.76 KDM4E (0.75) SMN1; SMN2KDM4ELMNAALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-121574323-A Dibenzothiophene sulfonyl covalent organic framework material and application thereof in thiadiazole and derivative photocatalytic synthesis 三峡大学 2026-02-27 CN disclosed
US-20210346369-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC. (US) 2021-11-11 US disclosed
CN-100432070-C Novel sulfamides and their use as endothelin receptor antagonists ACTELION PHARMACEUTICALS LTD (CH) 2008-11-12 CN disclosed
US-7285549-B2 Sulfamides and their use as endothelin receptor antagonists ACTELION PHARMACEUTICALS LTD. (CH) 2007-10-23 US disclosed
US-7285549-B2 Sulfamides and their use as endothelin receptor antagonists ACTELION PHARMACEUTICALS LTD. (CH) 2007-10-23 US disclosed
US-7285549-B2 Sulfamides and their use as endothelin receptor antagonists ACTELION PHARMACEUTICALS LTD. (CH) 2007-10-23 US disclosed
EP-1693372-A1 Novel Sulfamides and their use as endothelin receptor antagonists Actelion Pharmaceuticals Ltd. (CH) 2006-08-23 EP disclosed
US-7094781-B2 Sulfamides and their use as endothelin receptor antagonists ACTELION PHARMACEUTICALS LTD. (CH) 2006-08-22 US disclosed
US-20060178365-A1 Optionally oxidized 6-(2-(5-methylthio-2-pyrimidinyloxy)ethoxy)-2-phenylpyrimidin-4-yl-substituted sulfamides BOLLI MARTIN 2006-08-10 US disclosed
EP-1345920-B1 NOVEL SULFAMIDES AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2006-04-12 EP disclosed
CN-1524079-A Novel sulfonamides and their use as endothelin receptor antagonists ������˹ҩƷ��˾ 2004-08-25 CN disclosed
US-20040077670-A1 Novel sulfamides and their use as endothelin receptor antagonists ACTELION PHARMACEUTICALS LTD. (CH) 2004-04-22 US disclosed
EP-1345920-A1 NOVEL SULFAMIDES AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS Actelion Pharmaceuticals Ltd. (CH) 2003-09-24 EP disclosed
WO-2002053557-A1 NOVEL SULFAMIDES AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2002-07-11 WO disclosed
EP-0170057-B1 PROCESS FOR THE PREPARATION OF N-PHENYL(PYRIDYL) SULFONYL DIAMIDES BASF Aktiengesellschaft (DE) 1987-01-14 EP disclosed
EP-0170057-A2 Process for the preparation of N-phenyl(pyridyl) sulfonyl diamides BASF Aktiengesellschaft (DE) 1986-02-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210346369-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES BAX, BCL2, BCL3 TSHR 3610/4885ATM 1331/4885SMN1; SMN2 3576/4885
US-20060178365-A1 Optionally oxidized 6-(2-(5-methylthio-2-pyrimidinyloxy)ethoxy)-2-phenylpyrimidin-4-yl-substituted sulfamides EDNRA, EDNRB, ECE2 TSHR 1351/4885ATM 4221/4885SMN1; SMN2 1494/4885
US-20040077670-A1 Novel sulfamides and their use as endothelin receptor antagonists EDNRA, EDNRB, ECE1 TSHR 481/4885ATM 4263/4885SMN1; SMN2 2976/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.